| Assay Method Information | |
| | ChEMBL_2123272 (CHEMBL4832505) |
| Description: | Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as beta-arrestin recruitment by measuring U50,488 EC50 at 10 uM using furimazine as a substrate pretreated for 5 mins followed by ligand addition coincubation with U50,488 measured for 35 mins by BRET assay |
| Affinity data for this assay | |
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