Assay Method Information

Assay Name:  ChEMBL_757154 (CHEMBL1803294)
Description:  Antagonist activity at human GnRH receptor expressed in CHO cells assessed as inhibition of GnRH-induced arachidonic acid release using [5,6,8,9,11,12,14,15-3H]arachidonic acid preincubated for 15 mins measured after 45 mins by scintillation counting in presence of 40% human serum
Affinity data for this assay
 

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