Assay Method Information

Assay Name:  ChEMBL_1933658 (CHEMBL4479310)
Description:  Antagonist activity at human P2X7 receptor in LPS/IFN-gamma-differentiated human THP-1 cells assessed as suppression of BzATP-stimulated IL-1beta release per-incubated for 30 mins before BzATP addition and measured after 30 mins by ELISA
Affinity data for this assay
 

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