Assay Method Information | |
| ChEMBL_1784658 (CHEMBL4256175) |
Description: | Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated for 5 mins followed by (+/-)-epibatidine addition measured for 78 secs by Fluo-4-AM dye based FLIPR assay |
Affinity data for this assay | |
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