Assay Method Information

Assay Name:  ChEMBL_1718151 (CHEMBL4133151)
Description:  Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins followed by ATP addition measured after 20 mins by spectrofluorometric analysis
Affinity data for this assay
 

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