Assay Method Information | |
| ChEMBL_1718151 (CHEMBL4133151) |
Description: | Antagonist activity at human P2X7 receptor expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins followed by ATP addition measured after 20 mins by spectrofluorometric analysis |
Affinity data for this assay | |
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