| Assay Method Information | |
| | ChEMBL_2123256 (CHEMBL4832489) |
| Description: | Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as inhibition of forskolin induced cAMP production by measuring U50,488 EC50 at 10 uM pretreated for 30 mins followed by coincubation with U50,488 measured after 30 mins by HTRF assay |
| Affinity data for this assay | |
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