Assay Method Information

Assay Name:  ChEMBL_1698014 (CHEMBL4048904)
Description:  Antagonist activity at human SP/Myc epitope-tagged dopamine D4 receptor expressed in HEK293T cells assessed as inhibition of dopamine-induced RLuc8-fused Galphai1 activation preincubated for 15 mins followed by dopamine induction measured after 2 mins by BRET assay
Affinity data for this assay
 

If you find an error in this entry please send us an E-mail