Assay Method Information

Assay Name:  ChEMBL_2213976 (CHEMBL5127108)
Description:  Inverse agonist activity at 6His-tagged human RORC LBD (262 to 507 residues) expressed in Escherichia coli BL21 (DE3) cells assessed as inhibition of N-terminal biotinylated SRC1-4 derived QKPTSGPQTPQAQQKSLLQQLLTE coactivator peptide by luminescence based AlphaScreen analysis
Affinity data for this assay
 

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