| Assay Method Information | |
| | ChEMBL_1883062 (CHEMBL4384561) |
| Description: | Antagonist activity at human DEF3-RLuc fused CXCR4 receptor expressed in HEK293T cells co-expressing DEF3-Beta-arrestin-2-mVenus assessed as inhibition of CXCL12-induced beta-arrestin2 recruitment preincubated for 60 mins followed by CXCL12 addition measured after 20 mins by BRET assay |
| Affinity data for this assay | |
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