Assay Method Information

Assay Name:  ChEMBL_1830178 (CHEMBL4330052)
Description:  Inhibition of full length human N-terminal FLAG-tagged HDAC8 (1 to 377 residues) expressed in HEK293 cells preincubated for 15 mins followed by Boc-[trifluoroacetyl-Lys]-AMC substrate addition measured after 30 mins by fluorimetric method
Affinity data for this assay
 

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