Assay Method Information

Assay Name:  ChEMBL_1780734 (CHEMBL4252251)
Description:  Antagonist activity at human P2X7R expressed in HEK293 cells assessed as inhibition of ATP-induced ethidium iodide uptake preincubated for 10 mins followed by ATP induction measured after 25 mins by fluorescence assay
Affinity data for this assay
 

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