Assay Method Information

Assay Name:  ChEMBL_1711201 (CHEMBL4121250)
Description:  Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium flux preincubated for 20 mins followed by AVP addition measured for 5 mins by Fluo-4-AM dye based FLIPR assay
Affinity data for this assay
 

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