Assay Method Information | |
| ChEMBL_1711201 (CHEMBL4121250) |
Description: | Antagonist activity at human liver vasopressin V1a receptor expressed in CHO cells assessed as inhibition of agonist-induced intracellular calcium flux preincubated for 20 mins followed by AVP addition measured for 5 mins by Fluo-4-AM dye based FLIPR assay |
Affinity data for this assay | |
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