| Assay Method Information | |
| | titration assay |
| Description: | To identify inhibitors of TMPRSS2 that may be used directly in clinical studies or as lead compounds to develop targeted drugs, we screened several chemical libraries with active TMPRSS2 protease, the chromogenic TMPRSS2 peptide substrate Boc-Gln-Ala-Arg-MCA, and compound concentrations of 5 μmol/L. We have used a similar approach to identify inhibitors of the hepsin protease. |
| Affinity data for this assay | |
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