| Assay Method Information | |
| | ChEMBL_815799 (CHEMBL2025966) |
| Description: | Antagonist activity at human alpha4beta2 nAChR expressed in SH-EP1 cells assessed as inhibition of carbamylcholine induced 86Rb+ ion efflux preincubated for 10 mins prior to carbamylcholine-induction measured after 5 mins by flip-plate technique |
| Affinity data for this assay | |
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