| Assay Method Information | |
| | ChEMBL_2649823 |
| Description: | Antagonist activity at wild type HA-tagged human GnRH1 receptor expressed in HEK293T cells assessed as inhibition of GnRH peptide-stimulated IP1 accumulation by measuring GnRH peptide EC50 at 100 uM pretreated for 1 hr followed by stimulation with GnRH peptide for 1 hr (Rvb = 2.5 nM) |
| Affinity data for this assay | |
|---|---|
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