Assay Method Information | |
| ChEMBL_2171278 (CHEMBL5056412) |
Description: | Inhibition of human recombinant CYP2D6 expressed in insect microsome using (3-[2-(N,N-dimethyl-N-methylammonium)-ethyl]-7-methoxy-4-methylcoumarin iodide as a substrate incubated for 30 mins followed by addition of NADPH regenerating system measured immediately by fluorescence based analysis |
Affinity data for this assay | |
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