| Assay Method Information | |
| | ChEMBL_1878648 (CHEMBL4380042) |
| Description: | Inverse agonist activity at human N-terminal His6-tagged RORgammat LBD (265 to 518 residues) expressed in Escherichia coli BL21 (DE3) assessed as inhibition of N-terminal biotinylated co-activator SRC1 box2 peptide recruitment measured after 30 mins by TR-FRET assay |
| Affinity data for this assay | |
|---|---|
| If you find an error in this entry please send us an E-mail | |