Assay Method Information

Assay Name:  ChEMBL_956568 (CHEMBL2380018)
Description:  Antagonist activity at human adenosine A1 receptor expressed in CHOK1 cells assessed as inhibition of R-PIA/forskolin-induced cAMP accumulation incubated for 15 mins prior to R-PIA/forskolin challenge measured after 5.5 to 6 hrs by beta-galactosidase reporter gene assay
Affinity data for this assay
 

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