Assay Method Information

Assay Name:  ChEMBL_1784656 (CHEMBL4256173)
Description:  Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated for 5 mins followed by (+/-)-epibatidine addition measured for 78 secs by Fluo-4-AM dye based FLIPR assay
Affinity data for this assay
 

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