| Assay Method Information | |
| | ChEMBL_1736349 (CHEMBL4151885) |
| Description: | Inverse agonist activity at biotinylated HN-Avi-MBP-TCS-human RORgammat (258 to 518 residues) assessed as inhibition of biotinylated SRC-1 peptide NCOA1 (677 to 700 residues) recruitment incubated with coactivator peptide 15 mins before enzyme addition and further incubated for 1 hr by HTRF-FRET assay |
| Affinity data for this assay | |
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