Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 3313
TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286100(US9517228, Example 1 (4'S) | US9987253, Example 1 ...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
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TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM397087(US9987253, Example 2 | US10617673, Example 2 | US1...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286104(US9517228, Example 3 (2S,4′S) | US9987253, E...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286106(US9517228, Example 4 (2S,4′S) | US9987253, E...)
Affinity DataIC50: 100nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286105(US9517228, Example 3a (2S,4′R) | US9987253, ...)
Affinity DataIC50: 550nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286101(US9517228, Example 1a (4'R) | US9987253, Example 1...)
Affinity DataIC50: 5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286103(US9517228, Example 2a | US9987253, Example 2a | US...)
Affinity DataIC50: 5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Jenrin Discovery

US Patent
LigandPNGBDBM286107(US9517228, Example 4a (2S,4′R) | US9987253, ...)
Affinity DataIC50: 5.50E+3nMAssay Description:Compound binding to CB1R was assessed in competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain....More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/25/2020
Entry Details
Go to US Patent