Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 3202
TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394126(US9975861, 6)
Affinity DataIC50: 4.34E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394127(US9975861, 9)
Affinity DataIC50: 6.93E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 7.11E+3nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 8.13E+3nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 1.26E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 1.26E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 1.57E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394123(US9975861, 3 | US9975861, 5 | US9975861, 4)
Affinity DataIC50: 1.61E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394126(US9975861, 6)
Affinity DataIC50: 3.68E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394122(US9975861, 2)
Affinity DataIC50: 4.07E+4nMAssay Description:Human recombinant GSK-3β was purchased from Millipore (Millipore Iberica S.A.U.) The prephosphorylated polypeptide substrate was purchased from ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Fondazione Istituto Itaiano Di Tecnologia

US Patent
LigandPNGBDBM394122(US9975861, 2)
Affinity DataIC50: 5.03E+4nMAssay Description:β-secretase (BACE-1, Sigma-Aldrich) inhibition studies were performed by employing a peptide mimicking APP sequence as substrate (Methoxycoumari...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/10/2020
Entry Details
Go to US Patent