Compile Data Set for Download or QSAR
Report error Found 63 Enz. Inhib. hit(s) with all data for entry = 3042
TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389576(US9951029, 75 | N-{6-bromo-2-[(E)-2-(4- methoxyphe...)
Affinity DataIC50: 74nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389583(US9951029, 83 | N-{2-[(E)-2-(4- methoxyphenyl)viny...)
Affinity DataIC50: 134nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389615(US9951029, 132 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 246nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389591(US9951029, 100 | N'-{2-[(E)-2-(4- isopropylphenyl)...)
Affinity DataIC50: 258nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389604(US9951029, 121 | N,N-dimethyl-N'-(2-{(E)-2-[4- (me...)
Affinity DataIC50: 326nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389608(US9951029, 125 | N'-{6-chloro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 412nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389616(US9951029, 133 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 440nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389586(US9951029, 88 | N,N-dimethyl-N'-(2-{(E)-2-[4- (met...)
Affinity DataIC50: 461nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389611(US9951029, 128 | N'-{6-fluoro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 582nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389574(US9951029, 68 | N'-{2-[(E)-2-(4- fluorophenyl)viny...)
Affinity DataIC50: 811nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389613(US9951029, 130 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 873nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389612(US9951029, 129 | N,N-diethyl-N'-{6-fluoro-2-[(E)-2...)
Affinity DataIC50: 874nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389585(US9951029, 85 | N,N-dimethyl-N'-{2-[(E)-2-(2- thie...)
Affinity DataIC50: 950nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389610(US9951029, 127 | N'-{6-fluoro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 1.26E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389602(US9951029, 112 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 1.26E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389606(US9951029, 123 | N'-{6-chloro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 1.27E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389559(US9951029, 7 | N'-{6-bromo-2-[(E)-2-(4- methoxyphe...)
Affinity DataIC50: 1.39E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389609(US9951029, 126 | N'-{6-chloro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 1.40E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389558(US9951029, 6 | N'-{6-bromo-2-[(E)-2-(4- methoxyphe...)
Affinity DataIC50: 1.42E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389590(US9951029, 99 | N,N-diethyl-N'-{2-[(E)-2-(4- isopr...)
Affinity DataIC50: 1.51E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389603(US9951029, 119 | N,N-dimethyl-N'-(2-{(E)-2-[4- (me...)
Affinity DataIC50: 1.51E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389562(US9951029, 15 | N'-{6-bromo-2-[(E)-2-(4- fluorophe...)
Affinity DataIC50: 1.55E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389582(US9951029, 82 | N,N-dimethyl-N'-{2-[(E)-2-(2- thie...)
Affinity DataIC50: 1.64E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389581(US9951029, 81 | N'-{6-chloro-2-[(E)-2-(3,4- difluo...)
Affinity DataIC50: 1.70E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389578(US9951029, 77 | N,N-diethyl-N'-(2-{(E)-2-[4- (meth...)
Affinity DataIC50: 1.76E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389554(US9951029, 1 | N'-{6-chloro-2-[(E)-2-(4- methoxyph...)
Affinity DataIC50: 1.91E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389560(US9951029, 11 | N'-{6-bromo-2-[(E)-2-(4- methoxyph...)
Affinity DataIC50: 1.96E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389614(US9951029, 131 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 1.98E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389573(US9951029, 57 | N'-{6-bromo-2-[(E)-2-(3,4- difluor...)
Affinity DataIC50: 2.00E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389589(US9951029, 98 | N'-{2-[(E)-2-(4- isopropylphenyl)v...)
Affinity DataIC50: 2.02E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389575(US9951029, 69 | N,N-diethyl-N'-{2-[(E)-2-(4- fluor...)
Affinity DataIC50: 2.12E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389567(US9951029, 21 | N'-{6-chloro-2-[(E)-2-(4- fluoroph...)
Affinity DataIC50: 2.26E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389565(US9951029, 18 | N'-{6-bromo-2-[(E)-2-(4- fluorophe...)
Affinity DataIC50: 2.28E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389595(US9951029, 104 | N'-{6-chloro-2-[(E)-2-(2- thienyl...)
Affinity DataIC50: 2.31E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389584(US9951029, 84 | N,N-diethyl-N'-{2-[(E)-2-(2- thien...)
Affinity DataIC50: 2.33E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389599(US9951029, 109 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 2.39E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389566(US9951029, 20 | N'-{6-chloro-2-[(E)-2-(4- fluoroph...)
Affinity DataIC50: 2.39E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389594(US9951029, 103 | N'-{6-chloro-2-[(E)-2-(2- thienyl...)
Affinity DataIC50: 2.93E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389607(US9951029, 124 | N'-{6-chloro-2-[(E)-2-(4- isoprop...)
Affinity DataIC50: 2.97E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389563(US9951029, 16 | N'-{2-[(E)-2-(4- fluorophenyl)viny...)
Affinity DataIC50: 3.08E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389588(US9951029, 93 | N'-{2-[(E)-2-(3,4- difluorophenyl)...)
Affinity DataIC50: 3.25E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389577(US9951029, 76 | N-[3-({6-bromo-2-[(E)-2-(4- methox...)
Affinity DataIC50: 3.70E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389605(US9951029, 122 | 2-{(E)-2-[4- (methylsulfonyl)phen...)
Affinity DataIC50: 3.82E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389568(US9951029, 22 | N'-{6-fluoro-2-[(E)-2-(4- fluoroph...)
Affinity DataIC50: 4.20E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389579(US9951029, 78 | N,N-dimethyl-N'-(2-{(E)-2-[4- (met...)
Affinity DataIC50: 4.50E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389569(US9951029, 23 | N,N-diethyl-N'-{6-fluoro-2-[(E)-2-...)
Affinity DataIC50: 4.76E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389561(US9951029, 12 | N'-{2-[(E)-2-(4- methoxyphenyl)vin...)
Affinity DataIC50: 5.11E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389600(US9951029, 110 | N'-(6-chloro-2-{(E)-2-[4- (methyl...)
Affinity DataIC50: 5.62E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389598(US9951029, 108 | N,N-dimethyl-N'-{2-[(E)-2-(2- thi...)
Affinity DataIC50: 6.29E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
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TargetReceptor-type tyrosine-protein kinase FLT3(Human)
Vichem Chemie Kutató

US Patent
LigandPNGBDBM389580(US9951029, 79 | N'-{6-chloro-2-[(E)-2-(3,4- difluo...)
Affinity DataIC50: 6.32E+3nMAssay Description:FLT3(ITD) biochemical assays were performed on two different assay system platforms, using Transcreener ADP Assay FP method (BellBrook Labs, Madison,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/16/2020
Entry Details
Go to US Patent

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