Compile Data Set for Download or QSAR
Report error Found 93 Enz. Inhib. hit(s) with all data for entry = 2435
LigandPNGBDBM365304(US9868720, No. 425 | (2-Methoxy-4-methyl- phenyl)-...)
Affinity DataKi:  0.170nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365250(US9868720, No. 169 | [6-(1-Methyl-piperidin- 4-yl)...)
Affinity DataKi:  0.400nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365305(US9868720, No. 426 | {3-[2-(3,3-Difluoro- pyrroli...)
Affinity DataKi:  0.5nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365231(US9868720, No. 65 | [2-(2-Methyl-pyrrolidin- 1-yl)...)
Affinity DataKi:  0.735nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365240(US9868720, No. 111 | [2-((R)-2-Methyl-pyrrolidin- ...)
Affinity DataKi:  0.850nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365260(US9868720, No. 202 | (4-Cyclopropyl-pyridin- 2-yl)...)
Affinity DataKi:  0.950nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365261(US9868720, No. 402 | 2-Imidazol-1-yl-1-{3-[2- (2-m...)
Affinity DataKi:  1.59nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365290(US9868720, No. 376 | (1-Methyl-1H-imidazol- 4-yl)-...)
Affinity DataKi:  1.72nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365252(US9868720, No. 175 | 1-{4-[2-((R)-2-Methyl- pyrrol...)
Affinity DataKi:  2.20nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM50059205(CHEMBL3393322 | US9868720, No. 92)
Affinity DataKi:  2.43nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365237(US9868720, No. 96 | [2-(3,3-Difluoro-piperidin- 1-...)
Affinity DataKi:  3.10nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365259(US9868720, No. 201 | [2-(3,3-Difluoro-pyrrolidin- ...)
Affinity DataKi:  3.20nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365248(US9868720, No. 160 | [2-(3,3-Difluoro-pyrrolidin- ...)
Affinity DataKi:  4.42nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365232(US9868720, No. 66 | (2-Pyrrolidin-1-yl-6-pyr- roli...)
Affinity DataKi:  4.80nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365298(US9868720, No. 404 | {2-(3,3-Difluoro-pyrrolidin- ...)
Affinity DataKi:  4.92nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365302(US9868720, No. 423 | {2-(1-Methyl-1H-pyrazol- 4-yl...)
Affinity DataKi:  5.21nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365281(US9868720, No. 332 | 1-Methyl-4-[2-(2-methyl- pyrr...)
Affinity DataKi:  6.12nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365261(US9868720, No. 402 | 2-Imidazol-1-yl-1-{3-[2- (2-m...)
Affinity DataKi:  7.69nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365253(US9868720, No. 177 | 3-{4-[2-(2-Methyl-pyrrolidin-...)
Affinity DataKi:  8.03nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365258(US9868720, No. 200 | (4-tert-Butyl-pyridin-2- yl)-...)
Affinity DataKi:  8.34nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365242(US9868720, No. 120 | (4-Chloro-pyridin-2-yl)- [2-(...)
Affinity DataKi:  8.55nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365292(US9868720, No. 388 | {2-(2-Methyl-2H-pyrazol- 3-yl...)
Affinity DataKi:  8.75nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365293(US9868720, No. 391 | [2-Cyclopentyl-6-(1- oxetan-3...)
Affinity DataKi:  9nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365245(US9868720, No. 143 | [2-((2R,5R)-2,5-Dimethyl- pyr...)
Affinity DataKi:  10.4nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365289(US9868720, No. 375 | 1-{3-[2-((R)-2-Methyl- pyrrol...)
Affinity DataKi:  11.1nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365238(US9868720, No. 105 | 4-[2-(3,3-Difluoro-pyr- rolid...)
Affinity DataKi:  11.7nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365303(US9868720, No. 424 | 1-{4-[2-(1-Methyl-1H- pyrazol...)
Affinity DataKi:  12.4nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365227(US9868720, No. 47 | 2-{Methyl-[4-pyrrolidin- 3-yl-...)
Affinity DataKi:  12.6nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365243(US9868720, No. 125 | (4-Methoxy-pyridin-2-yl)- [2-...)
Affinity DataKi:  15.2nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365249(US9868720, No. 161 | 3-Oxo-3-{4-[2-pyrrolidin- 1-y...)
Affinity DataKi:  15.3nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365241(US9868720, No. 112 | [2-((S)-2-Methyl-pyrrolidin- ...)
Affinity DataKi:  15.8nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365306(US9868720, No. 427 | N-(4-chloropyridin-2-yl)- 2-(...)
Affinity DataKi:  16nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365280(US9868720, No. 331 | 1-Methyl-5-[2-((R)-2- methyl-...)
Affinity DataKi:  18.4nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365223(US9868720, No. 24 | (4-Methyl-pyridin-2-yl)- (6-pi...)
Affinity DataKi:  20.5nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365218(US9868720, No. 7 | 1-(3-(2-(1-methyl-1H-pyrazol-4-...)
Affinity DataKi:  20.7nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365282(US9868720, No. 348 | [2-(2-Ethyl-morpholin- 4-yl)-...)
Affinity DataKi:  22.6nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365299(US9868720, No. 407 | [2-Cyclobutyl-6-(1-oxetan- 3-...)
Affinity DataKi:  26nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365266(US9868720, No. 250 | 1-{4-[2-(3,4-Difluoro- pyrrol...)
Affinity DataKi:  26.7nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365254(US9868720, No. 178 | 1-{3-[2-(3,3-Difluoro- pyrrol...)
Affinity DataKi:  26.8nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365247(US9868720, No. 156 | 1-Acetyl-4-[2-(3,3- difluoro-...)
Affinity DataKi:  26.9nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365288(US9868720, No. 374 | [6-(1-Methanesulfonyl- azetid...)
Affinity DataKi:  30.6nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365239(US9868720, No. 106 | 1-{3-[6-(4-Methyl-pyridin- 2-...)
Affinity DataKi:  30.7nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365279(US9868720, No. 330 | [6-(1-Methanesulfonyl- piperi...)
Affinity DataKi:  31.8nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365276(US9868720, No. 307 | {2-(3,3-Difluoro-azetidin- 1-...)
Affinity DataKi:  31.9nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365291(US9868720, No. 385 | [2-Cyclopentyl-6-(1- methanes...)
Affinity DataKi:  36.8nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365251(US9868720, No. 173 | 3-{3-[2-Cyclopropyl-6- (4-tri...)
Affinity DataKi:  37nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365256(US9868720, No. 184 | Cyclopropyl-{3-[2-(3,3- diflu...)
Affinity DataKi:  41.5nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365262(US9868720, No. 206 | 1-{4-[6-(4-Trifluoromethyl- p...)
Affinity DataKi:  43.3nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365268(US9868720, No. 252 | [2-(3,4,6,7-Tetrahydro- imida...)
Affinity DataKi:  43.5nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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LigandPNGBDBM365222(US9868720, No. 22 | (4-Fluoro-phenyl)-{3-[2- methy...)
Affinity DataKi:  43.6nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2019
Entry Details
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