Compile Data Set for Download or QSAR
Report error Found 321 Enz. Inhib. hit(s) with all data for entry = 2072
TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354359(2-((2-ethyl-6-(4-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354376(2-(4-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354377(2-(4-(2-ethyl-3-((4- (4-fluorophenyl)-5- (2,2,2- t...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354395((S)-(1-(3- (dimethylamino) propylsulfonyl)- 4-(2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354481(2-((2-ethyl-6-(3- morpholino- pvrrolidin-1- yl)imi...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354492(2-((2-ethyl-6-(4- ((2-oxooxazolidin- 5- yl)methyl)...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354499(2-((6-(7-acetoyl- 2,7- diazaspiro[4.4] nonan-2-yl)...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354500(methyl (1-(3-((5- cyano-4-(4- fluorophenyl) thiazo...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354501(N-((1-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354506((S)-2-((2-ethyl-6- (3-(2-(3- hydroxyazetidin-1- yl...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354507((S)-2-(1-(3-((5- cyano-4-(4- fluorophenyl) thiazol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354508((R)-2-((2-ethyl-6- (3-(2-(3- hydroxyazetidin-1- yl...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354509((R)-2-(1(3-((5- cyano-4-(4- fluorophenyl) thiazol-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354511(2-((2-ethyl-6-(3-(4- (hydroxymethyl) piperidin-1- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354512(2-((6-(3-(4- acetoylpiperazin-1- yl)pyrrolidin-1-y...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354513(N-(1-(1-(3-((5- cyano-4-(4- fluorophenyl) thiazol-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354514(2-((2-ethyl-6-(3-(4- hydroxypiperidin- 1-yl)pyrrol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354515(2-((2-ethyl-6-(3-(4- methoxypiperidin- 1-yl)pyrrol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354516(2-((2-ethyl-6- ((3S,4S)-3- hydroxy-4- morpholino- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354520(2-((6-(3- aminoazetidin-1- yl)-2- ethylimidazo[1,2...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354521(2-((2-ethyl-6-(3-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354522(N-(1-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354543(2-((2-ethyl-6-(1-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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TargetAutotaxin(Human)
Galapagos

US Patent
LigandPNGBDBM354544(2-(6-((2-ethyl-6-(1- (2-(3- hydroxyazetidin-1- yl)...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a fluorescent hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using the fluorogenic autotax...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354337(2-((6-(4-(2- (azetidin-1-yl)-2- oxoethyl)piperazin...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354338(2-(4-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354339((R)-2-((2-ethyl-6- (4-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

LigandPNGBDBM354340((S)-2-((2-ethyl-6- (4-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354341(2-((2-ethyl-6-(4-(2- oxo-2-(pyrrolidin- 1- yl)ethy...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

LigandPNGBDBM354342(2-(4-(3-((5-cyano- 4-(4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

LigandPNGBDBM354343(2-((2-ethyl-6-(4-(2- morpholino-2- oxoethyl)pipera...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354344(2-((2-ethyl-6-(4-(2- (3-fluoroazetidin-1- yl)-2- o...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354345(2-((2-ethyl-6-(4-(2- (3-hydroxyazetidin- 1-yl)acet...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354353(2-((2-ethyl-6-(1-(2- (3-hydroxyazetidin- 1-yl)-2-o...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354355(2-((2-ethyl-6-(1-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354356((R)-2-((2-ethyl-6- (1-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354357((S)-2-((2-ethyl-6- (1-(2-(3- hydroxypyrrolidin- 1-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354358(2-(4-(2-ethyl-3-((4- (4- fluorophenl) thiazol-2- y...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

LigandPNGBDBM354359(2-((2-ethyl-6-(4-(2- (3-hydroxyazetidin- 1-yl)-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354361(2-(4-(2-ethyl-3-((4- (4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354365((R)-2-(4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354366((S)-2-(4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354372(5-((4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol-2-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354374(2-(4-(2-ethyl-3-((4- (4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354375(2-(4-(2-ethyl-3-((4- (4-fluorophenyl)-5- (hydroxym...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354377(2-(4-(2-ethyl-3-((4- (4-fluorophenyl)-5- (2,2,2- t...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
Go to US Patent

LigandPNGBDBM354378(1-(2-(4-(2-ethyl-3- ((4-(4- fluorophenyl) thiazol-...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354379((4-(2-ethyl-3-((4- (4- fluorophenyl) thiazol-2- yl...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354380(N-(2-ethyl-6-(4- ((tetrahydrofuran-2- yl)methyl)pi...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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LigandPNGBDBM354381(3-(4-(2-ethyl-3-((4- (4- fluorophenyl) thiazol-2- ...)
Affinity DataIC50: 55nMAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate.5 μL of a dil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2019
Entry Details
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