Compile Data Set for Download or QSAR
Report error Found 132 Enz. Inhib. hit(s) with all data for entry = 1871
LigandPNGBDBM50071821(CHEMBL3410872 | US9783573, Example 6)
Affinity DataIC50: 3nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
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Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50030280(CHEMBL3339214 | US9783573, Example 10)
Affinity DataIC50: 3nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345152(US9783573, Example 2)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345168(US9783573, Example 18)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345172((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50030270(CHEMBL3339219 | US9783573, Example 23)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345175((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345205(US9783573, Example 55)
Affinity DataIC50: 4nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345176((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 5nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345213(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 5nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345171((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345207(US9783573, Example 57)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345215(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 6nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345209(N1-((35,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 7nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345205(US9783573, Example 55)
Affinity DataIC50: 9nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50030270(CHEMBL3339219 | US9783573, Example 23)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345207(US9783573, Example 57)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345214(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 10nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345163(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345170(US9783573, Example 20)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345209(N1-((35,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 11nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345161(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345163(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345206(US9783573, Example 56)
Affinity DataIC50: 12nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345172((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345214(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345215(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 14nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50071821(CHEMBL3410872 | US9783573, Example 6)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345175((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50030278(CHEMBL3339215 | US9783573, Example 38)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345211(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 16nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345171((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345206(US9783573, Example 56)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345213(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 17nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345161(N1-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 18nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345208(US9783573, Example 58)
Affinity DataIC50: 18nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345204(N4-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 21nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345199(US9783573, Example 49)
Affinity DataIC50: 22nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345210(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 22nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM50030280(CHEMBL3339214 | US9783573, Example 10)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345168(US9783573, Example 18)
Affinity DataIC50: 23nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345201(N4-((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino...)
Affinity DataIC50: 27nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
Go to US Patent

LigandPNGBDBM345208(US9783573, Example 58)
Affinity DataIC50: 27nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345152(US9783573, Example 2)
Affinity DataIC50: 28nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345211(N1-((3S,5S)-1-((S)-3,3-Dimethyl-2-((S)-2- (methyla...)
Affinity DataIC50: 31nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345174((S)-2-((S)-3,3-Dimethyl-2-((S)-2-(methylamino) pro...)
Affinity DataIC50: 33nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR2-3 (125-356, C...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345182(US9783573, Example 32)
Affinity DataIC50: 35nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345170(US9783573, Example 20)
Affinity DataIC50: 37nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of His-BIR3 (241-356, XIA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345180(US9783573, Example 30)
Affinity DataIC50: 38nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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LigandPNGBDBM345202((S)-2-((S)-3,3-Dimethyl-2-((S)-2- (methylamino)pro...)
Affinity DataIC50: 42nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3 (241-356...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2019
Entry Details
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