Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 136
LigandPNGBDBM187126(US9670181, 6 4-(dibenzo[b,d]furan-2-ylmethyl)-1-et...)
Affinity DataIC50: 0.120nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187169(US9670181, 50 4-((2-(ethylamino)-6-methoxyquinolin...)
Affinity DataIC50: 0.280nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187210(US9670181, 86 4-((6-ethoxy-2-(ethylamino)-7-fluoro...)
Affinity DataIC50: 0.300nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187169(US9670181, 50 4-((2-(ethylamino)-6-methoxyquinolin...)
Affinity DataIC50: 0.340nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187209(US9670181, 85 1-ethyl-6,7-dimethoxy-4-((6-methoxyq...)
Affinity DataIC50: 0.400nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187160(US9670181, 40 1-ethyl-4-((2-(ethylamino)-6-methoxy...)
Affinity DataIC50: 0.400nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187162(US9670181, 42 1-ethyl-6,7-dimethoxy-4-((6-methoxy-...)
Affinity DataIC50: 0.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187127(US9670181, 7 4-(dibenzo[b,d]furan-2-ylmethyl)-6,7-...)
Affinity DataIC50: 0.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187174(US9670181, 53 4-((2-(isopropylamino)-6-methoxyquin...)
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187126(US9670181, 6 4-(dibenzo[b,d]furan-2-ylmethyl)-1-et...)
Affinity DataIC50: 0.900nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187184(US9670181, 62 6,7-dimethoxy-4-((6-(methylamino)-[1...)
Affinity DataIC50: 1.10nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187186(US9670181, 64 4-((6-(ethylamino)-[1,3]dioxolo[4,5-...)
Affinity DataIC50: 1.20nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187206(US9670181, 82 1-ethyl-4-((2-(ethylamino)-7-fluoro-...)
Affinity DataIC50: 1.40nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187155(US9670181, 35 4-((2-(ethylamino)-6-methylquinolin-...)
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187192(US9670181, 69 N-(2-((3-((1-ethyl-3-hydroxy-6,7-dim...)
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187173(US9670181, 52 6,7-dimethoxy-4-((6-methoxy-2-(propy...)
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187208(US9670181, 84 6,7-dimethoxy-4-((6-methoxyquinolin-...)
Affinity DataIC50: 1.60nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187159(US9670181, 39 1-ethyl-6,7-dimethoxy-4-((6-methoxy-...)
Affinity DataIC50: 1.60nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187212(US9670181, 88 N-(2-((6-ethoxy-3-((3-hydroxy-6,7-di...)
Affinity DataIC50: 1.80nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187189(US9670181, 67 4-((2-(ethylamino)-6-methoxyquinolin...)
Affinity DataIC50: 1.80nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187154(US9670181, 34 6,7-dimethoxy-4-((6-methyl-2-(methyl...)
Affinity DataIC50: 1.90nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187201(US9670181, 77 1-ethyl-6,7-dimethoxy-4-((6-methoxy-...)
Affinity DataIC50: 2nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187182(US9670181, 61 1-ethyl-6,7-dimethoxy-4-((6-(methyla...)
Affinity DataIC50: 2.20nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187200(US9670181, 76 6,7-dimethoxy-4-((6-methoxy-2-((2-me...)
Affinity DataIC50: 2.30nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187193(US9670181, 70 4-((2-(ethylamino)-7-fluoro-6-methox...)
Affinity DataIC50: 2.40nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
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LigandPNGBDBM187158(US9670181, 38 6,7-dimethoxy-4-((6-methoxy-2-(propy...)
Affinity DataIC50: 2.70nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187181(US9670181, 60 6,7-dimethoxy-1-methyl-4-((6-(methyl...)
Affinity DataIC50: 2.70nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187197(US9670181, 73 N-(2-((3-((3-hydroxy-6,7-dimethoxy-1...)
Affinity DataIC50: 2.70nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187204(US9670181, 80 6,7-dimethoxy-4-((2-methylquinolin-6...)
Affinity DataIC50: 3.20nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187163(US9670181, 43 1-ethyl-4-((2-(isopropylamino)-6-met...)
Affinity DataIC50: 3.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187211(US9670181, 87 N-(2-((6-(cyclopropylmethoxy)-3-((1-...)
Affinity DataIC50: 3.90nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187152(US9670181, 32 6,7-dimethoxy-4-((7-methoxyquinolin-...)
Affinity DataIC50: 4nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187176(US9670181, 55 N-(2-((3-((3-hydroxy-6,7-dimethoxy-1...)
Affinity DataIC50: 4.40nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187170(US9670181, 49 4-((6-ethoxy-2-(ethylamino)quinolin-...)
Affinity DataIC50: 4.60nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187161(US9670181, 41 4-((6-ethoxy-2-(ethylamino)quinolin-...)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187157(US9670181, 37 6,7-dimethoxy-4-((6-methoxy-2-(methy...)
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187148(US9670181, 28 4-((5-ethoxyquinolin-3-yl)methyl)-6,...)
Affinity DataIC50: 6nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187198(US9670181, 74 6,7-dimethoxy-1-propyl-4-(quinolin-3...)
Affinity DataIC50: 6.10nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187205(US9670181, 81 1-ethyl-6,7-dimethoxy-4-((2-methylqu...)
Affinity DataIC50: 7.5nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187164(US9670181, 44 4-((2-(benzylamino)-6-methoxyquinoli...)
Affinity DataIC50: 8nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187207(US9670181, 83 N-(2-((6-(cyclopropylmethoxy)-3-((3-...)
Affinity DataIC50: 10nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187139(US9670181, 19 1-ethyl-6,7-dimethoxy-4-(naphthalen-...)
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187167(US9670181, 47 4-((2-(ethylamino)-6-methoxyquinolin...)
Affinity DataIC50: 11nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187153(US9670181, 33 6,7-dimethoxy-1-methyl-4-((6-methyl-...)
Affinity DataIC50: 13nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187151(US9670181, 31 1-ethyl-6,7-dimethoxy-4-((7-methoxyq...)
Affinity DataIC50: 13nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187137(US9670181, 17 6,7-dimethoxy-1-methyl-4-(naphthalen...)
Affinity DataIC50: 14nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
Entry Details
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LigandPNGBDBM187188(US9670181, 66 4-((2-ethyl-6-methoxyquinolin-3-yl)m...)
Affinity DataIC50: 16nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
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LigandPNGBDBM187147(US9670181, 27 6,7-dimethoxy-4-((5-methoxyquinolin-...)
Affinity DataIC50: 17nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
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LigandPNGBDBM187150(US9670181, 30 4-((7-ethoxyquinolin-3-yl)methyl)-6,...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
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Date in BDB:
5/19/2018
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LigandPNGBDBM187175(US9670181, 54 6,7-dimethoxy-4-((6-methoxy-2-((2,2,...)
Affinity DataIC50: 23nMpH: 7.4 T: 2°CAssay Description:The PDE assay is based on the homogenous time-resolved fluorescence resonance energy transfer (TR-FRET) technology (LANCE from Perkin Elmer). This co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
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