Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 1105
TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309987(US9657003, 186 | N-((S)-1-(3-(3-chloro-4-cyano-2-m...)
Affinity DataIC50: 11nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309988(US9657003, 206 | (S)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataIC50: 29nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309990(US9657003, 222 | (R)-N-(2-(3-(4-cyano-3,5-difluoro...)
Affinity DataIC50: 33nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309973(US9657003, 32 | (S)-N-(1-(3-(4-cyano-3-methylpheny...)
Affinity DataIC50: 34nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309995(US9657003, 338 | (S)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataIC50: 42nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309992(US9657003, 249 | (S)-N-{1-[3-(3-Chloro-4-cyano-5-f...)
Affinity DataIC50: 42nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309981(US9657003, 91 | (S)-N-(1-(3-(3-chloro-4-cyanopheny...)
Affinity DataIC50: 54nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309982(US9657003, 94 | (S)-N-(1-(3-(3-chloro-4-cyanopheny...)
Affinity DataIC50: 57nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309983(US9657003, 103 | N-((R)-1-(3-(3-chloro-4-cyanophen...)
Affinity DataIC50: 71nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309980(US9657003, 53 | N-(2-(3-(4-cyano-3-methylphenyl)-1...)
Affinity DataIC50: 88nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309986(US9657003, 132 | (R)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataIC50: 93nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309979(US9657003, 56 | N-((S)-1-(3-(3-chloro-4-cyanopheny...)
Affinity DataIC50: 96nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309993(US9657003, 324 | (S)-N-(1-(3-(3-chloro-4-cyano-5-f...)
Affinity DataIC50: 128nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309985(US9657003, 124 | N-((S)-1-(3-(3-chloro-4-cyanophen...)
Affinity DataIC50: 133nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309989(US9657003, 219 | (S)-3-acetyl-N-(2-(3-(4-cyano-3,5...)
Affinity DataIC50: 146nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309978(US9657003, 52 | N-(2-(3-(3,4-dicyanophenyl)-1H-pyr...)
Affinity DataIC50: 149nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309976(US9657003, 34 | (S)-3-acetyl-N-(1-(3-(3-chloro-4-c...)
Affinity DataIC50: 172nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309991(US9657003, 248 | (S)-N-{1-[3-(3-Chloro-4-cyanophen...)
Affinity DataIC50: 190nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309994(US9657003, Bicalutamide)
Affinity DataIC50: 228nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309972(US9657003, 8 | N-(2-(5-(3,4-dichlorophenyl)furan-2...)
Affinity DataIC50: 606nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309987(US9657003, 186 | N-((S)-1-(3-(3-chloro-4-cyano-2-m...)
Affinity DataKi:  3nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309973(US9657003, 32 | (S)-N-(1-(3-(4-cyano-3-methylpheny...)
Affinity DataKi:  6nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309982(US9657003, 94 | (S)-N-(1-(3-(3-chloro-4-cyanopheny...)
Affinity DataKi:  8nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309990(US9657003, 222 | (R)-N-(2-(3-(4-cyano-3,5-difluoro...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309988(US9657003, 206 | (S)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataKi:  12nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309981(US9657003, 91 | (S)-N-(1-(3-(3-chloro-4-cyanopheny...)
Affinity DataKi:  13nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309995(US9657003, 338 | (S)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309979(US9657003, 56 | N-((S)-1-(3-(3-chloro-4-cyanopheny...)
Affinity DataKi:  14nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309992(US9657003, 249 | (S)-N-{1-[3-(3-Chloro-4-cyano-5-f...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309976(US9657003, 34 | (S)-3-acetyl-N-(1-(3-(3-chloro-4-c...)
Affinity DataKi:  16nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309983(US9657003, 103 | N-((R)-1-(3-(3-chloro-4-cyanophen...)
Affinity DataKi:  17nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309980(US9657003, 53 | N-(2-(3-(4-cyano-3-methylphenyl)-1...)
Affinity DataKi:  18nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309993(US9657003, 324 | (S)-N-(1-(3-(3-chloro-4-cyano-5-f...)
Affinity DataKi:  25nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309978(US9657003, 52 | N-(2-(3-(3,4-dicyanophenyl)-1H-pyr...)
Affinity DataKi:  27nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309986(US9657003, 132 | (R)-N-(1-(3-(3-chloro-4-cyanophen...)
Affinity DataKi:  29nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309991(US9657003, 248 | (S)-N-{1-[3-(3-Chloro-4-cyanophen...)
Affinity DataKi:  31nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309985(US9657003, 124 | N-((S)-1-(3-(3-chloro-4-cyanophen...)
Affinity DataKi:  38nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309989(US9657003, 219 | (S)-3-acetyl-N-(2-(3-(4-cyano-3,5...)
Affinity DataKi:  40nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309994(US9657003, Bicalutamide)
Affinity DataKi:  40nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent

TargetAndrogen receptor(Human)
Orion

US Patent
LigandPNGBDBM309972(US9657003, 8 | N-(2-(5-(3,4-dichlorophenyl)furan-2...)
Affinity DataKi:  62nMAssay Description:Androgen receptor (AR) binding affinities of test compounds were studied in cytosolic lysates obtained from ventral prostates of castrated rats by co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/9/2019
Entry Details
Go to US Patent