Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 1086
TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116303(US8637504, 81 | US9273053, 81 | US9650371, 81)
Affinity DataIC50: 7nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116274(US9270353, 16 | US8637504, 16 | US9650371, 16)
Affinity DataIC50: 10nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116304(US8637504, 99 | US9273053, 99 | US9650371, 99)
Affinity DataIC50: 14nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116288(US8637504, 51 | US9273053, 51 | US9650371, 51)
Affinity DataIC50: 16nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM308068(Compound 200 | US9650371, 21)
Affinity DataIC50: 19nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116292(US8637504, 59 | US9273053, 59 | US9650371, 59)
Affinity DataIC50: 19nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116305(US8637504, 101 | US9273053, 101 | US9650371, 101)
Affinity DataIC50: 22nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116302(US8637504, 79 | US9273053, 79 | US9650371, 79)
Affinity DataIC50: 24nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116297(US8637504, 70 | US9273053, 70 | US9650371, 70)
Affinity DataIC50: 36nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116306(US8637504, 102 | US9273053, 102 | US9650371, 102)
Affinity DataIC50: 36nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116279(US8637504, 24 | US9273053, 24 | US9650371, 24)
Affinity DataIC50: 54nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116301(US8637504, 76 | US9273053, 76 | US9650371, 76)
Affinity DataIC50: 62nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116307(US8637504, 104 | US9273053, 104 | US9650371, 104)
Affinity DataIC50: 63nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM308072(US9650371, 33)
Affinity DataIC50: 73nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116289(US8637504, 53 | US9273053, 53 | US9650371, 53)
Affinity DataIC50: 76nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116286(US8637504, 47 | US9273053, 47 | US9650371, 47)
Affinity DataIC50: 91nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM308067(Intermediate Compound (147) | US9650371, 20)
Affinity DataIC50: 95nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116281(US8637504, 35 | US9650371, 35)
Affinity DataIC50: 96nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116283(US8637504, 39 | US9273053, 39 | US9650371, 39)
Affinity DataIC50: 97nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116308(US8637504, 106 | US9273053, 106 | US9650371, 106)
Affinity DataIC50: 102nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116294(US8637504, 61 | US9273053, 61 | US9650371, 61)
Affinity DataIC50: 169nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116291(US8637504, 58 | US9273053, 58 | US9650371, 58)
Affinity DataIC50: 186nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116299(US8637504, 73 | US9273053, 73 | US9650371, 73)
Affinity DataIC50: 234nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116293(US8637504, 60 | US9273053, 60 | US9650371, 60)
Affinity DataIC50: 243nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116298(US8637504, 72 | US9273053, 72 | US9650371, 72)
Affinity DataIC50: 250nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116287(US8637504, 48 | US9273053, 48 | US9650371, 48)
Affinity DataIC50: 273nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116296(US8637504, 66 | US9273053, 66 | US9650371, 66)
Affinity DataIC50: 296nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116282(US8637504, 38 | US9273053, 38 | US9650371, 38)
Affinity DataIC50: 304nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116290(US8637504, 56 | US9273053, 56 | US9650371, 56)
Affinity DataIC50: 352nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116295(US8637504, 63 | US9273053, 63 | US9650371, 63)
Affinity DataIC50: 435nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116272(US8637504, 2 | US9273053, 2 | US9650371, 2)
Affinity DataIC50: 514nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
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TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116277(US8637504, 22 | US9273053, 22 | US9650371, 22)
Affinity DataIC50: 572nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116285(US8637504, 46 | US9273053, 46 | US9650371, 46)
Affinity DataIC50: 611nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116300(US8637504, 75 | US9273053, 75 | US9650371, 75)
Affinity DataIC50: 697nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116273(US8637504, 3 | US9273053, 3 | US9650371, 3)
Affinity DataIC50: 966nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116284(US8637504, 44 | US9273053, 44 | US9650371, 44)
Affinity DataIC50: 2.13E+3nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent

TargetBeta-secretase 1(Human)
Shionogi

US Patent
LigandPNGBDBM116278(US8637504, 23 | US9273053, 23 | US9650371, 23)
Affinity DataIC50: 5.28E+3nMAssay Description:48.5 uL of substrate peptide solution (Biotin-XSEVNLDAEFRHDSGC-Eu: X=ε-amino-n-capronic acid, Eu=Europium cryptate) was added to each well of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/3/2019
Entry Details
Go to US Patent