Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 1188
LigandPNGBDBM312090(US9603889, Example 2)
Affinity DataIC50: 30nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM50030266(CHEMBL3339223 | US9603889, Example 8)
Affinity DataIC50: 30nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312102(US9603889, Example 13 | (S)-N-Benzyl-2- ((S)-3,3- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312103(US9603889, Example 14 | (S)-2-((S)- 3,3-Dimethyl- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312129(US9603889, Example 40)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312121(US9603889, Example 32 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312099(US9603889, Example 10)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM50030266(CHEMBL3339223 | US9603889, Example 8)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312127(US9603889, Example 38)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312130(US9603889, Example 41)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312114(US9603889, Example 25 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312113(US9603889, Example 24 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312091(US9603889, Example 3)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM50030268(CHEMBL3339221 | US9603889, Example 1)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312094(US9603889, Example 6)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312131(US9603889, Example 42)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312100(US9603889, Example 11 | (S)-N-(2,3- Dichlorobenzyl...)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312105(US9603889, Example 16 | (S)-2-((S)-3,3- Dimethyl- ...)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312128(US9603889, Example 39)
Affinity DataIC50: 80nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM50030268(CHEMBL3339221 | US9603889, Example 1)
Affinity DataIC50: 90nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312104(US9603889, Example 15 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312116(US9603889, Example 27 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312101(US9603889, Example 12 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312125(US9603889, Example 36 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312115(US9603889, Example 26 | (3S)-N-(1-(2- Chlorophenyl...)
Affinity DataIC50: 100nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312092(US9603889, Example 4)
Affinity DataIC50: 100nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312106(US9603889, Example 17 | N1-(((S)-2-((S)- 3,3-dimet...)
Affinity DataIC50: 100nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312130(US9603889, Example 41)
Affinity DataIC50: 110nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312111(US9603889, Example 22 | (S)-2-((S)-3,3- Dimethyl- ...)
Affinity DataIC50: 110nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312109(US9603889, Example 20 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 110nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312122(US9603889, Example 33 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312091(US9603889, Example 3)
Affinity DataIC50: 120nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312112(US9603889, Example 23 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312107(US9603889, Example 18 | (S)-N-((S)-1-(3- Chlorophe...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312097(US9603889, Example 9)
Affinity DataIC50: 130nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312113(US9603889, Example 24 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 130nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312132(US9603889, Example 43)
Affinity DataIC50: 150nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312094(US9603889, Example 6)
Affinity DataIC50: 150nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312123(US9603889, Example 34 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312118(US9603889, Example 29 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312117(US9603889, Example 28 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312112(US9603889, Example 23 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 170nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312132(US9603889, Example 43)
Affinity DataIC50: 180nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312092(US9603889, Example 4)
Affinity DataIC50: 180nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312107(US9603889, Example 18 | (S)-N-((S)-1-(3- Chlorophe...)
Affinity DataIC50: 190nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312095(US9603889, Example 7)
Affinity DataIC50: 190nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312115(US9603889, Example 26 | (3S)-N-(1-(2- Chlorophenyl...)
Affinity DataIC50: 190nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312127(US9603889, Example 38)
Affinity DataIC50: 220nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
Go to US Patent

LigandPNGBDBM312093(US9603889, Example 5)
Affinity DataIC50: 220nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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LigandPNGBDBM312126(US9603889, Example 37 | N1-(((S)-2- ((S)-3,3- Dime...)
Affinity DataIC50: 230nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
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