Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 844
TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294083(US9585879, 52 | 6-Bromo-N′-dodecanoyl-1-ethy...)
Affinity DataIC50: 2.01E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294091(US9585879, 60 | 7-Chloro-N′-dodecanoyl-1-eth...)
Affinity DataIC50: 2.48E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM50384798(CHEMBL2037482 | US9585879, 6 | US9757369, 6)
Affinity DataIC50: 2.85E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294072(US9585879, 15 | 7-Chloro-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 3.12E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294087(US9585879, 56 | 6-Chloro-N′-dodecanoyl-1-eth...)
Affinity DataIC50: 3.18E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294078(US9585879, 47 | 6-Bromo-N′-dodecanoyl-4-hydr...)
Affinity DataIC50: 3.54E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294079(US9585879, 48 | 6-Chloro-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 3.81E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294089(US9585879, 58 | 7-Chloro-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 4.03E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294081(US9585879, 50 | 6-Bromo-N′-dodecanoyl-4-hydr...)
Affinity DataIC50: 4.28E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294070(US9585879, 13 | N′-Dodecanoyl-4-hydroxy-2-ox...)
Affinity DataIC50: 4.47E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294090(US9585879, 59 | 7-Chloro-1-ethyl-4-hydroxy-N′...)
Affinity DataIC50: 4.83E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294076(US9585879, 45 | 1-(cyclopropylmethyl)-N′-dod...)
Affinity DataIC50: 5.25E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(US9585879, 46 | 1-Benzyl-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 5.51E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294073(US9585879, 17 | 6-Fluoro-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 5.81E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294085(US9585879, 54 | 6-Chloro-N′-dodecanoyl-4-hyd...)
Affinity DataIC50: 5.95E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294092(US9585879, 61 | 1-Benzyl-7-chloro-4-hydroxy-N̸...)
Affinity DataIC50: 5.96E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294093(US9585879, 62 | 1-Benzyl-7-chloro-N′dodecano...)
Affinity DataIC50: 5.99E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294080(US9585879, 49 | 6-Bromo-4-hydroxy-1-methyl-N′...)
Affinity DataIC50: 6.28E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294088(US9585879, 57 | 7-Chloro-4-hydroxy-1-methyl-N̸...)
Affinity DataIC50: 6.66E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294094(US9585879, 63 | N′,1-Dibenzyl-N′-dodec...)
Affinity DataIC50: 6.84E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294074(US9585879, 42 | 4-Hydroxy-1-(isoprenyl)-N′-o...)
Affinity DataIC50: 7.11E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294082(US9585879, 51 | 6-Bromo-1-ethyl-4-hydroxy-N′...)
Affinity DataIC50: 7.34E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294068(US9585879, 4 | N′-Dodecanoyl-4-hydroxy-1-met...)
Affinity DataIC50: 7.35E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294075(US9585879, 43 | N′-Dodecanoyl-4-hydroxy-1-(i...)
Affinity DataIC50: 7.78E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294084(US9585879, 53 | 6-Chloro-4-hydroxy-1-methyl-N̸...)
Affinity DataIC50: 8.48E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294067(US9585879, 3 | 4-Hydroxy-1-methyl-N′-octanoy...)
Affinity DataIC50: 8.67E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294071(US9585879, 14 | 7-Chloro-4-hydroxy-N′-octano...)
Affinity DataIC50: 9.00E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent

TargetGlycogen synthase kinase-3 beta(Human)
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294086(US9585879, 55 | 6-Chloro-1-ethyl-4-hydroxy-N′...)
Affinity DataIC50: 9.42E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2019
Entry Details
Go to US Patent