Compile Data Set for Download or QSAR
Report error Found 358 Enz. Inhib. hit(s) with all data for entry = 683
TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286684BDBM286684(7-((R)-3-Amino-pyrrolidin-1-ylmethyl)-3-(5-chloro-...)
Affinity DataIC50: 7.90nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286640BDBM286640(7-((R)-3-Amino-pyrrolidin-1-ylmethyl)-8-bromo-3-(5...)
Affinity DataIC50: 9.80nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286685BDBM286685(US9567304, Compound B-20 | 3-(5-Chloro-2-ethanesul...)
Affinity DataIC50: 11nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286641BDBM286641(7-((S)-3-Aminomethyl-pyrrolidin-1-ylmethyl)-8-brom...)
Affinity DataIC50: 12nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286724BDBM286724(7-((S)-3- Aminomethyl- pyrrolidin-1- ylmethyl)-6-b...)
Affinity DataIC50: 12nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286718BDBM286718(7-((R)-3-Amino-pyrrolidin-1-ylmethyl)-6-bromo-3-(5...)
Affinity DataIC50: 12nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286721BDBM286721(N-{(R)-1-[6-Bromo-3-(5-chloro-2-ethanesulfonyl-ben...)
Affinity DataIC50: 13nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286912BDBM286912(8-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((R...)
Affinity DataIC50: 14nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286687BDBM286687(3-(5-Chloro-2-ethanesulfonyl-benzyl)-7-((R)-3-meth...)
Affinity DataIC50: 15nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286586BDBM286586(7-((R)-3-Amino-piperidin-1-ylmethyl)-8-chloro-3-(5...)
Affinity DataIC50: 15nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286722BDBM286722(N-{(R)-1-[6-Bromo-3-(5-chloro-2-ethanesulfonyl-ben...)
Affinity DataIC50: 15nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286723BDBM286723(6-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((R...)
Affinity DataIC50: 15nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286719BDBM286719(6-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((R...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286574BDBM286574(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286672BDBM286672(3-(5-Chloro-2-ethanesulfonyl-benzyl)-7-piperazin-1...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286628BDBM286628(7-((S)-3-Amino-piperidin-1-ylmethyl)-8-chloro-3-(5...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286773BDBM286773(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286629BDBM286629(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286709BDBM286709(7-((R)-3-Amino-pyrrolidin-1-ylmethyl)-6-chloro-3-(...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286905BDBM286905(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286714BDBM286714(6-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-(4-...)
Affinity DataIC50: 16nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286630BDBM286630(7-((S)-2-Aminomethyl-pyrrolidin-1-ylmethyl)-8-chlo...)
Affinity DataIC50: 17nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286904BDBM286904(7-((S)-3-Aminomethyl-pyrrolidin-1-ylmethyl)-8-chlo...)
Affinity DataIC50: 17nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286953BDBM286953(7-[[(3R)-3-Aminopiperidin-1-yl]methyl]-8-chloro-3-...)
Affinity DataIC50: 17nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286633BDBM286633(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 17nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286522BDBM286522(3-(5-Chloro-2-ethanesulfonyl-benzyl)-7-(4-methyl-p...)
Affinity DataIC50: 17nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286913BDBM286913(N-{(R)-1-[8-Bromo-3-(5-chloro-2-ethanesulfonyl-ben...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286643BDBM286643(3-(8-Bromo-2, 4-dioxo-6-trifluoromethyl-1,4-dihydr...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286918BDBM286918(8-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((R...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286681BDBM286681(7-((S)-3-Amino-pyrrolidin-1-ylmethyl)-3-(5-chloro-...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286764BDBM286764(2-Amino-N-{(R)-1-[8-chloro-3-(5-chloro-2-ethanesul...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286782BDBM286782(7-((S)-3-Amino-pyrrolidin-1-ylmethyl)-8-chloro-3-(...)
Affinity DataIC50: 18nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286639BDBM286639(8-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((R...)
Affinity DataIC50: 19nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286929BDBM286929(6,8-Dibromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7...)
Affinity DataIC50: 19nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286754BDBM286754(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 19nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286689BDBM286689(7-((S)-3-Aminomethyl-pyrrolidin-1-ylmethyl)-3-(5-c...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286802BDBM286802(7-((R)-2-Aminomethyl-pyrrolidin-1-ylmethyl)-8-chlo...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286729BDBM286729(6-Bromo-3-(5- chloro-2- ethanesulfonyl- benzyl)-7-...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286540BDBM286540(7-((R)-3-Amino-pyrrolidin-1-ylmethyl)-8-chloro-3-(...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286830BDBM286830(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286702BDBM286702(3-(5-Chloro-2-ethanesulfonyl-benzyl)-7-((R)-3-dime...)
Affinity DataIC50: 20nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286846BDBM286846(US9567304, Compound F-122 | (S)-1-[8-Chloro-3- (5-...)
Affinity DataIC50: 21nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286787BDBM286787(8-Chloro-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-((...)
Affinity DataIC50: 21nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286504BDBM286504(3-(5-Chloro-2-ethanesulfonyl-benzyl)-7-(4-methyl-p...)
Affinity DataIC50: 21nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286957BDBM286957((3R)-1-[[8-Chloro-3-[(5-chloro-2-ethylsulfonylphen...)
Affinity DataIC50: 21nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286818BDBM286818(7-((R)-3-Aminomethyl-pyrrolidin-1-ylmethyl)-8-chlo...)
Affinity DataIC50: 22nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286899BDBM286899(7-((R)-2-Aminomethyl-pyrrolidin-1-ylmethyl)-8-chlo...)
Affinity DataIC50: 22nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286969BDBM286969(8-Chloro-3-[(5-chloro-2-ethylsulfonylphenyl)methyl...)
Affinity DataIC50: 22nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286730BDBM286730(6-Bromo-3-(5-chloro-2-ethanesulfonyl-benzyl)-7-(3-...)
Affinity DataIC50: 22nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetEpithelial discoidin domain-containing receptor 1(Human)
Chugai Seiyaku Kabushiki Kaisha

US Patent
LigandChemical structure of BindingDB Monomer ID 286829BDBM286829(7-((S)-3-Aminomethyl-piperidin-1-ylmethyl)-8-chlor...)
Affinity DataIC50: 22nMT: 2°CAssay Description:DDR1 binding activity was measured using the LanthaScreen(Registered trademark) Eu Kinase Binding Assay (manufactured by Life Technologies Corporatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

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