Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 8514
TargetSodium/glucose cotransporter 2(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US9505734, I-D1-6 | US10294259, Compound Table 3.2)
Affinity DataIC50: 0.690nMAssay Description:The IC50 value of the inhibition of the cocrystal of I-D1-6 and L-proline prepared in Example 138 on SGLT2 and SGLT1 is measured according to the met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Tianjin Institute of Pharmaceutical Research

US Patent
LigandPNGBDBM254941(US9505734, I-D1-6 | US10294259, Compound Table 3.2)
Affinity DataIC50: 259nMAssay Description:The IC50 value of the inhibition of the cocrystal of I-D1-6 and L-proline prepared in Example 138 on SGLT2 and SGLT1 is measured according to the met...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
Go to US Patent