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Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 8422
TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247344(US9447091, 131)
Affinity DataIC50: 1.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247340(US9447091, 112)
Affinity DataIC50: 1.80nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247357(US9447091, 241)
Affinity DataIC50: 2.90nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247334(US9447091, 49)
Affinity DataIC50: 3.40nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247361(US9447091, 220)
Affinity DataIC50: 3.40nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247328(US9447091, 22)
Affinity DataIC50: 3.80nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247354(US9447091, 190)
Affinity DataIC50: 4.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247333(US9447091, 47)
Affinity DataIC50: 7nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247348(US9447091, 152)
Affinity DataIC50: 7.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247360(US9447091, 281)
Affinity DataIC50: 9nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247363(US9447091, 294)
Affinity DataIC50: 9.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247336(US9447091, 70)
Affinity DataIC50: 10nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247356(US9447091, 217)
Affinity DataIC50: 10.4nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247327(US9447091, 5)
Affinity DataIC50: 12nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247345(US9447091, 133)
Affinity DataIC50: 14nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247358(US9447091, 244)
Affinity DataIC50: 14nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247353(US9447091, 178)
Affinity DataIC50: 14.9nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247338(US9447091, 82)
Affinity DataIC50: 16nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247331(US9447091, 30)
Affinity DataIC50: 16nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247364(US9447091, 319)
Affinity DataIC50: 18nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247355(US9447091, 204)
Affinity DataIC50: 20nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247330(US9447091, 26)
Affinity DataIC50: 21nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247335(US9447091, 69)
Affinity DataIC50: 22nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247350(US9447091, 158)
Affinity DataIC50: 22nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247337(US9447091, 72)
Affinity DataIC50: 32nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247362(US9447091, 289)
Affinity DataIC50: 32nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247332(US9447091, 38)
Affinity DataIC50: 33nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247329(US9447091, 25)
Affinity DataIC50: 34nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247339(US9447091, 83)
Affinity DataIC50: 37nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247366(US9447091, 259)
Affinity DataIC50: 45nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247347(US9447091, 142)
Affinity DataIC50: 48nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247352(US9447091, 170)
Affinity DataIC50: 59nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247342(US9447091, 123)
Affinity DataIC50: 61nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247349(US9447091, 155)
Affinity DataIC50: 62nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247343(US9447091, 127)
Affinity DataIC50: 62nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247365(US9447091, 322)
Affinity DataIC50: 65.8nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247341(US9447091, 119)
Affinity DataIC50: 83nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247359(US9447091, 280)
Affinity DataIC50: 90nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247351(US9447091, 169)
Affinity DataIC50: 94nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandPNGBDBM247346(US9447091, 134)
Affinity DataIC50: 98nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
Go to US Patent