Compile Data Set for Download or QSAR
Report error Found 75 Enz. Inhib. hit(s) with all data for entry = 8417
LigandPNGBDBM247218(US9434733, methyl 5-[[3-methyl-4-(4-oxo-7-tetrahyd...)
Affinity DataIC50: 8nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247206(US9434733, 2-[[3-[(4-fluorophenyl)methoxy]azetidin...)
Affinity DataIC50: 10nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247177(US9434733, 2-[4-methyl-1-[[4-(trifluoromethyl)phen...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247225(US9434733, 2-[1-[(5-chloro-2-thienyl)methyl]-4-met...)
Affinity DataIC50: 13nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247192(US9434733, 2-[1-[[4-(diethylamino)phenyl]methyl]-4...)
Affinity DataIC50: 13nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247183(US9434733, 2-[4-methyl-1-[[4-(trifluoromethoxy)phe...)
Affinity DataIC50: 19nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247195(US9434733, 2-[1-[(2-chloro-4-fluoro-phenyl)methyl]...)
Affinity DataIC50: 21nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247222(US9434733, 2-[(1R)-1-[3-(4-methoxyphenyl)azetidin-...)
Affinity DataIC50: 22nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247224(US9434733, 2-[4-methyl-1-[(5-methyl-2-thienyl)meth...)
Affinity DataIC50: 22nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247215(US9434733, 2-[1-[(3,4-difluorophenyl)methyl]-4-met...)
Affinity DataIC50: 23nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247186(US9434733, 2-[4-methyl-1-(quinoxalin-6-ylmethyl)py...)
Affinity DataIC50: 24nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247213(US9434733, 2-[1-[(5-fluoro-3-pyridyl)methyl]-4-met...)
Affinity DataIC50: 25nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247193(US9434733, 2-[1-(2-furylmethyl)-4-methyl-pyrrolidi...)
Affinity DataIC50: 25nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247196(US9434733, 2-[1-[(4-dimethylaminophenyl)methyl]-4-...)
Affinity DataIC50: 27nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247208(US9434733, 2-[4-methyl-1-[(5-methyl-2-furyl)methyl...)
Affinity DataIC50: 28nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247216(US9434733, 2-[1-[(4-chlorophenyl)methyl]-4-methyl-...)
Affinity DataIC50: 32nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247217(US9434733, 2-[1-[[6-(dimethylamino)-3-pyridyl]meth...)
Affinity DataIC50: 36nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247203(US9434733, 2-[4-methyl-1-(3-pyridylmethyl)pyrrolid...)
Affinity DataIC50: 37nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247185(US9434733, 2-[1-[(2-chloro-4-methoxy-phenyl)methyl...)
Affinity DataIC50: 41nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247207(US9434733, 2-[1-[3-(4-methoxyphenyl)azetidin-1-yl]...)
Affinity DataIC50: 47nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247197(US9434733, 2-[4-methyl-1-(p-tolylmethyl)pyrrolidin...)
Affinity DataIC50: 47nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
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LigandPNGBDBM247221(US9434733, 2-[(3R,4R)-1-[(2,4-difluorophenyl)methy...)
Affinity DataIC50: 47nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247181(US9434733, 2-[1-[(2,4-difluorophenyl)methyl]-4-met...)
Affinity DataIC50: 48nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247188(US9434733, 2-[1-[(4-methoxyphenyl)methyl]-4-methyl...)
Affinity DataIC50: 49nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247236(US9434733, 2-[1-benzyl-4-(trifluoromethyl)pyrrolid...)
Affinity DataIC50: 50nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247189(US9434733, 2-[4-methyl-1-(4-pyridylmethyl)pyrrolid...)
Affinity DataIC50: 52nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247227(US9434733, 2-(1-benzyl-4-methoxy-pyrrolidin-3-yl)-...)
Affinity DataIC50: 54nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247223(US9434733, 2-[1-[3-(4-fluorophenoxy)azetidin-1-yl]...)
Affinity DataIC50: 57nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247226(US9434733, 2-[4-methyl-1-[(4-pyrrolidin-1-ylphenyl...)
Affinity DataIC50: 61nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247204(US9434733, 2-[1-[(2,6-difluorophenyl)methyl]-4-met...)
Affinity DataIC50: 62nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247209(US9434733, 2-[1-[(5-chloro-2-furyl)methyl]-4-methy...)
Affinity DataIC50: 63nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247176(US9434733, 2-[1-[(6-methoxy-3-pyridyl)methyl]-4-me...)
Affinity DataIC50: 67nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247244(US9434733, 2-[1-[3-[(4-methoxyphenyl)methyl]azetid...)
Affinity DataIC50: 68nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247190(US9434733, 2-[[3-(4-fluorophenoxy)azetidin-1-yl]me...)
Affinity DataIC50: 80nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247233(US9434733, 2-[[3-[(4-methoxyphenoxy)methyl]azetidi...)
Affinity DataIC50: 82nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247233(US9434733, 2-[[3-[(4-methoxyphenoxy)methyl]azetidi...)
Affinity DataIC50: 82nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247239(US9434733, 2-[4-methoxy-1-[(4-methoxyphenyl)methyl...)
Affinity DataIC50: 83nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247238(US9434733, 2-[1-[3-(4-dimethylaminophenyl)azetidin...)
Affinity DataIC50: 86nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247202(US9434733, 2-[[3-(4-dimethylaminophenyl)azetidin-1...)
Affinity DataIC50: 86nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247175(US9434733, 7-(4-fluorophenyl)-2-[4-methyl-1-[[6-(t...)
Affinity DataIC50: 86nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247230(US9434733, 2-[4-methoxy-1-(p-tolylmethyl)pyrrolidi...)
Affinity DataIC50: 90nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247212(US9434733, 2-[[3-(4-methylphenoxy)azetidin-1-yl]me...)
Affinity DataIC50: 91nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247229(US9434733, 2-[1-[(4-fluorophenyl)methyl]-4-methoxy...)
Affinity DataIC50: 94nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247235(US9434733, 2-[1-[3-(4-pyrrolidin-1-ylphenyl)azetid...)
Affinity DataIC50: 110nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247232(US9434733, 2-[1-[3-(4-methylphenoxy)azetidin-1-yl]...)
Affinity DataIC50: 110nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247235(US9434733, 2-[1-[3-(4-pyrrolidin-1-ylphenyl)azetid...)
Affinity DataIC50: 110nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247232(US9434733, 2-[1-[3-(4-methylphenoxy)azetidin-1-yl]...)
Affinity DataIC50: 110nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247237(US9434733, 2-[[3-(5-pyrrolidin-1-ylpyrimidin-2-yl)...)
Affinity DataIC50: 120nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247228(US9434733, 2-[1-[3-(4-hydroxyphenyl)azetidin-1-yl]...)
Affinity DataIC50: 120nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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LigandPNGBDBM247210(US9434733, 2-[1-[3-(4-fluorophenyl)azetidin-1-yl]e...)
Affinity DataIC50: 128nMT: 2°CAssay Description:A PDE9 assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
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