Compile Data Set for Download or QSAR
Report error Found 144 Enz. Inhib. hit(s) with all data for entry = 8455
TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249396(US9434697, 108 | US9730931, Compound 108 | US10537...)
Affinity DataIC50: 0.200nMpH: 7.5 T: 2°CAssay Description:Recombinant FGFR1 (2.5 nM), or FGFR4 (12 nM) was prepared as a mixture with substrate KKKSPGEYVNIEFG (SEQ ID NO:1) (20 μM, FGFR1 substrate); Pol...More data for this Ligand-Target Pair
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Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249391(US9434697, 100 | US9730931, Compound 100 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
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Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249395(US9434697, 107 | US9730931, Compound 107 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249396(US9434697, 108 | US9730931, Compound 108 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249398(US9434697, 111 | US9730931, Compound 111 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249399(US9434697, 112 | US9730931, Compound 112 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249400(US9434697, 113 | US9730931, Compound 113 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
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Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249401(US9434697, 114 | US9730931, Compound 114 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
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Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249403(US9434697, 120 | US9730931, Compound 120 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249404(US9434697, 121 | US9730931, Compound 121 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249405(US9434697, 122 | US9730931, Compound 122 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249406(US9434697, 123 | US9730931, Compound 123 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249407(US9434697, 124 | US9730931, Compound 124 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249408(US9434697, 125 | US9730931, Compound 125 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249409(US9434697, 126 | US9730931, Compound 126 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249410(US9434697, 127 | US9730931, Compound 127 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249414(US9434697, 131 | US9730931, Compound 131 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249415(US9434697, 132 | US9730931, Compound 132 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249417(US9434697, 135 | US9730931, Compound 135 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249418(US9434697, 136 | US9730931, Compound 136 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249419(US9434697, 137 | US9730931, Compound 137 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249421(US9434697, 140 | US9730931, Compound 140 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249423(US9434697, 142 | US9730931, Compound 142 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249425(US9434697, 144 | US9730931, Compound 144 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249426(US9434697, 145 | US9730931, Compound 145 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249427(US9434697, 147 | US9730931, Compound 147 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249428(US9434697, 148 | US9730931, Compound 148 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249429(US9434697, 149 | US9730931, Compound 149 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249430(US9434697, 150 | US9730931, Compound 150 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249431(US9434697, 151 | US9730931, Compound 151 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249433(US9434697, 154 | US9730931, Compound 154 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249434(US9434697, 155 | US9730931, Compound 155 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249435(US9434697, 156 | US9730931, Compound 156 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249436(US9434697, 157 | US9730931, Compound 157 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249437(US9434697, 158 | US9730931, Compound 158 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249438(US9434697, 159 | US9730931, Compound 159 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249439(US9434697, 160 | US9730931, Compound 160 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249440(US9434697, 161 | US9730931, Compound 161 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249441(US9434697, 162 | US9730931, Compound 162 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249442(US9434697, 163 | US9730931, Compound 163 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249443(US9434697, 164 | US9730931, Compound 164 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249444(US9434697, 165 | US9730931, Compound 165 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249445(US9434697, 166 | US9730931, Compound 166 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249446(US9434697, 167 | US9730931, Compound 167 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249447(US9434697, 168 | US9730931, Compound 168 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249452(US9434697, 181 | US9730931, Compound 181 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249391(US9434697, 100 | US9730931, Compound 100 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
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US Patent
LigandPNGBDBM249396(US9434697, 108 | US9730931, Compound 108 | US10537...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
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US Patent
LigandPNGBDBM50355393(CHEMBL1834657 | US9434697, BGJ398 | US9730931, BGJ...)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:Recombinant FGFR1 (2.5 nM), or FGFR4 (12 nM) was prepared as a mixture with substrate KKKSPGEYVNIEFG (SEQ ID NO:1) (20 μM, FGFR1 substrate); Pol...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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PDB3D3D Structure (crystal)
TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM249413(US9434697, 130 | US9730931, Compound 130 | US10537...)
Affinity DataIC50: 2nMpH: 7.5 T: 2°CAssay Description:Compounds were profiled for FGFR inhibition activity at Reaction Biology Corporation (Malvern, Pa.) with their Kinase HotSpot assay. See, Anastassiad...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/18/2017
Entry Details
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