Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 8389
TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM50157531(US9428513, I-25 | CHEMBL3785917)
Affinity DataIC50: 9nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245805(US9428513, I-21)
Affinity DataIC50: 17nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245801(US9428513, I-17)
Affinity DataIC50: 18nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245800(US9428513, I-16)
Affinity DataIC50: 22nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245810(US9428513, I-27)
Affinity DataIC50: 26nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245797(US9428513, I-13)
Affinity DataIC50: 27nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245785(US9428513, I-1)
Affinity DataIC50: 32nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245787(US9428513, I-3)
Affinity DataIC50: 33nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245789(US9428513, I-5)
Affinity DataIC50: 33nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245806(US9428513, I-22)
Affinity DataIC50: 35nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245788(US9428513, I-4)
Affinity DataIC50: 43nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245812(US9428513, I-29)
Affinity DataIC50: 49nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245798(US9428513, I-14)
Affinity DataIC50: 49nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245790(US9428513, I-6)
Affinity DataIC50: 51nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245796(US9428513, I-12)
Affinity DataIC50: 51nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245794(US9428513, I-10)
Affinity DataIC50: 54nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245791(US9428513, I-7)
Affinity DataIC50: 55nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245792(US9428513, I-8)
Affinity DataIC50: 55nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245803(US9428513, I-19)
Affinity DataIC50: 58nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245808(US9428513, I-24)
Affinity DataIC50: 63nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245793(US9428513, I-9)
Affinity DataIC50: 65nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245802(US9428513, I-18)
Affinity DataIC50: 69nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245811(US9428513, I-28)
Affinity DataIC50: 69nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245807(US9428513, I-23)
Affinity DataIC50: 122nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245799(US9428513, I-15)
Affinity DataIC50: 123nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245809(US9428513, I-26)
Affinity DataIC50: 123nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245804(US9428513, I-20)
Affinity DataIC50: 157nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245786(US9428513, I-2)
Affinity DataIC50: 333nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
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TargetBromodomain-containing protein 4 [44-168](Human)
Boehringer Ingelheim International

US Patent
LigandPNGBDBM245795(US9428513, I-11)
Affinity DataIC50: 549nMAssay Description:Compounds are diluted in serial dilution 1:5 in assay buffer from 10 mM stock in DMSO (100 μM start concentration) in white OptiPlate-384 (PerkinE...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/28/2017
Entry Details
Go to US Patent