Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 8248
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238234(US9388210, 14a | US9388210, 6a)
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238243(US9388210, 16a)
Affinity DataIC50: 28nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238245(US9388210, 17a)
Affinity DataIC50: 53nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238238(US9388210, 15a | US9388210, 13a)
Affinity DataIC50: 56nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238234(US9388210, 14a | US9388210, 6a)
Affinity DataIC50: 128nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238238(US9388210, 15a | US9388210, 13a)
Affinity DataIC50: 474nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238235(US9388210, 14b | US9388210, 6b)
Affinity DataIC50: 501nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238244(US9388210, 16b)
Affinity DataIC50: 544nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238246(US9388210, 17b)
Affinity DataIC50: 605nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238236(US9388210, 6c)
Affinity DataIC50: 629nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238248(US9388210, 5b)
Affinity DataIC50: 770nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238247(US9388210, 5a)
Affinity DataIC50: 997nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238249(US9388210, 5c)
Affinity DataIC50: 1.02E+3nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
Go to US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238239(US9388210, 15b | US9388210, 13b)
Affinity DataIC50: 1.20E+3nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
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TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238237(US9388210, 6d)
Affinity DataIC50: 1.84E+3nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
Go to US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238235(US9388210, 14b | US9388210, 6b)
Affinity DataIC50: 2.03E+3nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
Go to US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rat)
Washington University

US Patent
LigandPNGBDBM238239(US9388210, 15b | US9388210, 13b)
Affinity DataIC50: 9.60E+3nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/17/2017
Entry Details
Go to US Patent