Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 7745
TargetSerine/threonine-protein kinase Sgk1(Mouse)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 26nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 2(Human)
Eli Lilly

US Patent
LigandPNGBDBM213821(US9296775, 1)
Affinity DataIC50: 6.10E+3nMpH: 7.5 T: 2°CAssay Description:The SGLT activity is measured as sodium-dependent 14C-AMG uptake in the above cell lines described as follows. One hundred uL of culture medium conta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2017
Entry Details
Go to US Patent