Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 7623
TargetMitogen-activated protein kinase 14(Human)
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LigandPNGBDBM206344(US9260410, 2)
Affinity DataIC50: 2.5nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
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TargetMitogen-activated protein kinase 14(Human)
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US Patent
LigandPNGBDBM206345(US9260410, 3)
Affinity DataIC50: 6.70nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
Entry Details
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TargetMitogen-activated protein kinase 14(Human)
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US Patent
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 12nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandPNGBDBM206345(US9260410, 3)
Affinity DataIC50: 18nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
Entry Details
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TargetMitogen-activated protein kinase 12(Human)
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US Patent
LigandPNGBDBM206345(US9260410, 3)
Affinity DataIC50: 146nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
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US Patent
LigandPNGBDBM206344(US9260410, 2)
Affinity DataIC50: 166nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
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Date in BDB:
12/28/2016
Entry Details
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TargetMitogen-activated protein kinase 12(Human)
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US Patent
LigandPNGBDBM206344(US9260410, 2)
Affinity DataIC50: 195nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 12(Human)
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US Patent
LigandPNGBDBM13533(1-[5-tert-butyl-2-(p-tolyl)pyrazol-3-yl]-3-[4-(2-m...)
Affinity DataIC50: 296nMAssay Description:The enzyme inhibitory activities of compounds disclosed herein were determined by fluorescence resonance energy transfer (FRET) using synthetic pepti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/28/2016
Entry Details
Go to US Patent