Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 7492
LigandPNGBDBM197718(US9216985, 1A)
Affinity DataIC50: 8nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
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LigandPNGBDBM197726(US9216985, 17A)
Affinity DataIC50: 8nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
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LigandPNGBDBM197724(US9216985, 15A)
Affinity DataIC50: 9nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197728(US9216985, 20A)
Affinity DataIC50: 10nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197722(US9216985, 10A)
Affinity DataIC50: 20nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197720(US9216985, 6A)
Affinity DataIC50: 20nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197721(US9216985, 7A)
Affinity DataIC50: 50nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197719(US9216985, 2A)
Affinity DataIC50: 80nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197725(US9216985, 16A)
Affinity DataIC50: 90nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197723(US9216985, 11A)
Affinity DataIC50: 110nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197727(US9216985, 19A)
Affinity DataIC50: 190nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197720(US9216985, 6A)
Affinity DataIC50: 300nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197728(US9216985, 20A)
Affinity DataIC50: 460nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197718(US9216985, 1A)
Affinity DataIC50: 650nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197724(US9216985, 15A)
Affinity DataIC50: 740nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197722(US9216985, 10A)
Affinity DataIC50: 740nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197728(US9216985, 20A)
Affinity DataIC50: 1.10E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197726(US9216985, 17A)
Affinity DataIC50: 1.20E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197718(US9216985, 1A)
Affinity DataIC50: 1.20E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197721(US9216985, 7A)
Affinity DataIC50: 1.30E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197719(US9216985, 2A)
Affinity DataIC50: 1.80E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197729(US9216985, 21A)
Affinity DataIC50: 2.10E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197723(US9216985, 11A)
Affinity DataIC50: 3.00E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197720(US9216985, 6A)
Affinity DataIC50: 3.10E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197726(US9216985, 17A)
Affinity DataIC50: 3.40E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197718(US9216985, 1A)
Affinity DataIC50: 3.70E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197719(US9216985, 2A)
Affinity DataIC50: 3.90E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197728(US9216985, 20A)
Affinity DataIC50: 4.10E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197727(US9216985, 19A)
Affinity DataIC50: 4.50E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197725(US9216985, 16A)
Affinity DataIC50: 5.40E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197721(US9216985, 7A)
Affinity DataIC50: 5.80E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197724(US9216985, 15A)
Affinity DataIC50: 7.30E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197724(US9216985, 15A)
Affinity DataIC50: 9.70E+3nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197729(US9216985, 21A)
Affinity DataIC50: 1.00E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197727(US9216985, 19A)
Affinity DataIC50: 1.00E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197727(US9216985, 19A)
Affinity DataIC50: 1.00E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197726(US9216985, 17A)
Affinity DataIC50: 1.00E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197725(US9216985, 16A)
Affinity DataIC50: 1.05E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197720(US9216985, 6A)
Affinity DataIC50: 1.50E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197721(US9216985, 7A)
Affinity DataIC50: 2.80E+4nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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LigandPNGBDBM197723(US9216985, 11A)
Affinity DataIC50: 1.15E+5nMAssay Description:The ability of the compounds of the present invention to inhibit the activity of four PI3K isoforms, PI3Kα, PI3Kβ, PI3Kγ, and PI3K&d...More data for this Ligand-Target Pair
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Date in BDB:
10/24/2016
Entry Details
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