Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 7346
TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190541(US9181185, 30b | US9624194, Compound 30b)
Affinity DataIC50: 130nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190556(US9181185, 6)
Affinity DataIC50: 152nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
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Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190558(US9181185, 8 | US9624194, Compound 8)
Affinity DataIC50: 193nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190561(US9181185, 19 | US9624194, Compound 19)
Affinity DataIC50: 244nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190559(US9181185, 14)
Affinity DataIC50: 246nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190553(US9181185, 30g | US9624194, Compound 30g)
Affinity DataIC50: 262nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190557(US9181185, 7 | US9624194, Compound 7)
Affinity DataIC50: 282nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190560(US9181185, 15 | US9624194, Compound 15)
Affinity DataIC50: 304nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190555(US9181185, 5 | US9624194, Compound 5)
Affinity DataIC50: 314nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190551(US9181185, 30f | US9624194, Compound 30f)
Affinity DataIC50: 376nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190542(US9181185, 31b | US9624194, Compound 31b)
Affinity DataIC50: 383nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190549(US9181185, 30e | US9624194, Compound 30e)
Affinity DataIC50: 461nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190550(US9181185, 31e | US9624194, Compound 31e)
Affinity DataIC50: 489nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190562(US9181185, 26 | US9624194, Compound 26)
Affinity DataIC50: 625nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190554(US9181185, 31g | US9624194, Compound 31g)
Affinity DataIC50: 690nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190545(US9181185, 30c | US9624194, Compound 30c)
Affinity DataIC50: 711nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190552(US9181185, 31f | US9624194, Compound 31f)
Affinity DataIC50: 804nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190547(US9181185, 30d | US9624194, Compound 30d)
Affinity DataIC50: 1.19E+3nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190543(US9181185, 30a | US9624194, Compound 30a)
Affinity DataIC50: 1.41E+3nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190548(US9181185, 31d | US9624194, Compound 31d)
Affinity DataIC50: 1.44E+3nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190546(US9181185, 31c | US9624194, Compound 31c)
Affinity DataIC50: 1.69E+3nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190544(US9181185, 31a | US9624194, Compound 31a)
Affinity DataIC50: 1.85E+3nMT: 2°CAssay Description:FLIPR or FLIPRTETRA Sodium Dye Assay with KCl and Test Article Pre-Incubation: Cells were prepared by plating the recombinant HEK293 cells or other h...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190561(US9181185, 19 | US9624194, Compound 19)
Affinity DataKi:  347nM ΔG°:  -38.4kJ/moleT: 2°CAssay Description:Cells: The hNav1.7 expressing HEK-293 cells were plated on 35 mm culture dishes pre-coated with poly-D-lysine in standard DMEM culture media (Mediate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190560(US9181185, 15 | US9624194, Compound 15)
Affinity DataKi:  917nM ΔG°:  -35.8kJ/moleT: 2°CAssay Description:Cells: The hNav1.7 expressing HEK-293 cells were plated on 35 mm culture dishes pre-coated with poly-D-lysine in standard DMEM culture media (Mediate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
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TargetSodium channel protein type 9 subunit alpha(Human)
Purdue Pharma

US Patent
LigandPNGBDBM190562(US9181185, 26 | US9624194, Compound 26)
Affinity DataKi:  2.26E+3nM ΔG°:  -33.5kJ/moleT: 2°CAssay Description:Cells: The hNav1.7 expressing HEK-293 cells were plated on 35 mm culture dishes pre-coated with poly-D-lysine in standard DMEM culture media (Mediate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2016
Entry Details
Go to US Patent