Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 7030
TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM47224(US9073917, 2-inventive)
Affinity DataIC50: 1nMAssay Description:The effect of the compounds of the invention on the activity of the enzyme PDE3 was evaluated by the company CEREP (Le bois I'Ev que, 86600 Celle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM47224(US9073917, 2-inventive)
Affinity DataIC50: 1nMAssay Description:The effect of the compounds of the invention on the activity of the enzyme PDE3 was evaluated by the company CEREP (Le bois I'Ev que, 86600 Celle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167515(US9073917, 12- comparative)
Affinity DataIC50: 3nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167510(US9073917, 7- comparative)
Affinity DataIC50: 3nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167506(US9073917, 1-inventive)
Affinity DataIC50: 4nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167515(US9073917, 12- comparative)
Affinity DataIC50: 4nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167510(US9073917, 7- comparative)
Affinity DataIC50: 4nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167507(US9073917, 4- comparative)
Affinity DataIC50: 6nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167506(US9073917, 1-inventive)
Affinity DataIC50: 6nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167508(US9073917, 5- comparative)
Affinity DataIC50: 6nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167512(US9073917, 11- comparative | US9073917, 9- compara...)
Affinity DataIC50: 8nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
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TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167513(US9073917, 10- comparative)
Affinity DataIC50: 9nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167516(US9073917, 13- comparative)
Affinity DataIC50: 10nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167516(US9073917, 13- comparative)
Affinity DataIC50: 11nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167509(US9073917, 6- comparative)
Affinity DataIC50: 13nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167512(US9073917, 11- comparative | US9073917, 9- compara...)
Affinity DataIC50: 15nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167511(US9073917, 8- comparative)
Affinity DataIC50: 21nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167513(US9073917, 10- comparative)
Affinity DataIC50: 22nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167508(US9073917, 5- comparative)
Affinity DataIC50: 23nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

LigandPNGBDBM167515(US9073917, 12- comparative)
Affinity DataIC50: 68nMAssay Description:The effect of the compounds of the invention on the activity of the enzyme PDE3 was evaluated by the company CEREP (Le bois I'Ev que, 86600 Celle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167507(US9073917, 4- comparative)
Affinity DataIC50: 72nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167511(US9073917, 8- comparative)
Affinity DataIC50: 102nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM167512(US9073917, 11- comparative | US9073917, 9- compara...)
Affinity DataIC50: 107nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167509(US9073917, 6- comparative)
Affinity DataIC50: 109nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM60452(US9073917, 3-comparative)
Affinity DataIC50: 900nMAssay Description:The effect of the compounds of the invention on the activity of the enzyme PDE3 was evaluated by the company CEREP (Le bois I'Ev que, 86600 Celle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase A(Human)
Sanofi

US Patent
LigandPNGBDBM167512(US9073917, 11- comparative | US9073917, 9- compara...)
Affinity DataIC50: 1.76E+3nMAssay Description:The capacity to inhibit the kinase activity of the enzyme is estimated by measuring the residual kinase activity of the enzyme in the presence of dif...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent

TargetAurora kinase B/Inner centromere protein(Human)
Sanofi

US Patent
LigandPNGBDBM60452(US9073917, 3-comparative)
Affinity DataIC50: 3.80E+3nMAssay Description:The effect of the compounds of the invention on the activity of the enzyme PDE3 was evaluated by the company CEREP (Le bois I'Ev que, 86600 Celle...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/29/2016
Entry Details
Go to US Patent