Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 6909
TargetAmine oxidase [flavin-containing] B(Human)
TBA

US Patent
LigandPNGBDBM10989((1R)-N-(prop-2-yn-1-yl)-2,3-dihydro-1H-inden-1-ami...)
Affinity DataIC50: 4nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
TBA

US Patent
LigandPNGBDBM158502(US9034303, Compound 3)
Affinity DataIC50: 20nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
TBA

US Patent
LigandPNGBDBM158501(US9034303, O-Methyl-M30)
Affinity DataIC50: 30nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
TBA

US Patent
LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50: 37nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
TBA

US Patent
LigandPNGBDBM36551(Chelator, M30 | US9034303, M30)
Affinity DataIC50: 57nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
TBA

US Patent
LigandPNGBDBM158502(US9034303, Compound 3)
Affinity DataIC50: 80nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] B(Human)
TBA

US Patent
LigandPNGBDBM158503(US9034303, Compound 4)
Affinity DataIC50: 100nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
TBA

US Patent
LigandPNGBDBM158503(US9034303, Compound 4)
Affinity DataIC50: 200nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
TBA

US Patent
LigandPNGBDBM158501(US9034303, O-Methyl-M30)
Affinity DataIC50: 275nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent

TargetAmine oxidase [flavin-containing] A(Human)
TBA

US Patent
LigandPNGBDBM10989((1R)-N-(prop-2-yn-1-yl)-2,3-dihydro-1H-inden-1-ami...)
Affinity DataIC50: 410nMAssay Description:MAO-A and MAO-B activity was measured using radioactive substrates. The substrate for MAO-A was 5 HT and for MAO-B was PEA. When measuring the activi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/23/2015
Entry Details
Go to US Patent