Compile Data Set for Download or QSAR
Report error Found 72 Enz. Inhib. hit(s) with all data for entry = 6769
TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152235BDBM152235(US8993552, 70)
Affinity DataIC50: 430nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent
PDB3D3D Structure (crystal)
TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152232BDBM152232(US8993552, 67)
Affinity DataIC50: 650nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152231BDBM152231(US8993552, 66)
Affinity DataIC50: 1.10E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152230BDBM152230(US8993552, 65)
Affinity DataIC50: 1.20E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152211BDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50: 1.20E+3nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152245BDBM152245(US8993552, 80)
Affinity DataIC50: 1.30E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152211BDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50: 1.90E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152211BDBM152211(BDBM152229 | US8993552, 1)
Affinity DataIC50: 1.90E+3nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152233BDBM152233(US8993552, 68)
Affinity DataIC50: 2.40E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152224BDBM152224(US8993552, 4)
Affinity DataIC50: 3.80E+3nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152247BDBM152247(US8993552, 82)
Affinity DataIC50: 4.40E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152236BDBM152236(US8993552, 71)
Affinity DataIC50: 4.60E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152237BDBM152237(US8993552, 72)
Affinity DataIC50: 4.80E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152241BDBM152241(US8993552, 76)
Affinity DataIC50: 6.30E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152249BDBM152249(US8993552, 32)
Affinity DataIC50: 7.00E+3nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152239BDBM152239(US8993552, 74)
Affinity DataIC50: 7.00E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152259BDBM152259(US8993552, 86)
Affinity DataIC50: 7.40E+3nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152242BDBM152242(US8993552, 77)
Affinity DataIC50: 8.70E+3nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 50302435BDBM50302435((4-(6-ethylthieno[2,3-d]pyrimidin-4-yl)piperazin-1...)
Affinity DataIC50: 1.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152251BDBM152251(US8993552, 34)
Affinity DataIC50: 1.20E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152243BDBM152243(US8993552, 78)
Affinity DataIC50: 1.20E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152228BDBM152228(US8993552, 63)
Affinity DataIC50: 1.20E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152249BDBM152249(US8993552, 32)
Affinity DataIC50: 1.30E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152234BDBM152234(US8993552, 69)
Affinity DataIC50: 1.60E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152227BDBM152227(US8993552, 61)
Affinity DataIC50: 2.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152244BDBM152244(US8993552, 79)
Affinity DataIC50: 2.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152238BDBM152238(US8993552, 73)
Affinity DataIC50: 2.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152248BDBM152248(US8993552, 83)
Affinity DataIC50: 2.70E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152250BDBM152250(US8993552, 33)
Affinity DataIC50: 2.80E+4nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152250BDBM152250(US8993552, 33)
Affinity DataIC50: 2.90E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152225BDBM152225(US8993552, 31)
Affinity DataIC50: 2.95E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152226BDBM152226(US8993552, 60)
Affinity DataIC50: 3.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152240BDBM152240(US8993552, 75)
Affinity DataIC50: 3.20E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152265BDBM152265(US8993552, 6G10_3 Compound 47)
Affinity DataIC50: 3.30E+4nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152252BDBM152252(US8993552, 35)
Affinity DataIC50: 3.50E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152213BDBM152213(US8993552, 3)
Affinity DataIC50: 3.50E+4nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152246BDBM152246(US8993552, 81)
Affinity DataIC50: 4.00E+4nMAssay Description:NMR spectroscopy validation of lead compounds. In embodiments of the present invention, and during development thereof, NMR spectroscopy: saturation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152212BDBM152212(US8993552, 2)
Affinity DataIC50: 4.20E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152219BDBM152219(US8993552, 15)
Affinity DataIC50: 4.90E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152222BDBM152222(US8993552, 21)
Affinity DataIC50: 5.00E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152261BDBM152261(US8993552, 4H8 Compound 42)
Affinity DataIC50: 5.00E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152214BDBM152214(US8993552, 8)
Affinity DataIC50: 6.00E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152253BDBM152253(US8993552, 36)
Affinity DataIC50: 6.30E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152265BDBM152265(US8993552, 6G10_3 Compound 47)
Affinity DataIC50: 6.70E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152220BDBM152220(US8993552, 16)
Affinity DataIC50: 7.10E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152258BDBM152258(US8993552, 85)
Affinity DataIC50: 7.20E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152272BDBM152272(US8993552, 6G10_14 Compound 58)
Affinity DataIC50: 8.00E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152213BDBM152213(US8993552, 3)
Affinity DataIC50: 8.30E+4nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152212BDBM152212(US8993552, 2)
Affinity DataIC50: 8.50E+4nMAssay Description:One potential limitation of the above FP assay is the risk of selection of compounds that may interfere with the FP assays and produce so called fals...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

TargetMenin(Human)
University of Michigan

US Patent
LigandChemical structure of BindingDB Monomer ID 152254BDBM152254(US8993552, 37)
Affinity DataIC50: 1.00E+5nMAssay Description:Assays effective in monitoring the inhibition of the MLL binding to menin were developed during experiments performed during the development of embod...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2015
Entry Details
US Patent

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