Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 6760
TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151195(US8987313, 36)
Affinity DataIC50: 100nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151194(US8987313, 35)
Affinity DataIC50: 100nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151197(US8987313, 42)
Affinity DataIC50: 110nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151187(US8987313, 11)
Affinity DataIC50: 120nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151193(US8987313, 32)
Affinity DataIC50: 120nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151196(US8987313, 39)
Affinity DataIC50: 130nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151191(US8987313, 25)
Affinity DataIC50: 140nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151194(US8987313, 35)
Affinity DataIC50: 150nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151199(US8987313, 24)
Affinity DataIC50: 150nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151201(US8987313, 31)
Affinity DataIC50: 150nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151185(US8987313, 5)
Affinity DataIC50: 160nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151189(US8987313, 18)
Affinity DataIC50: 160nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151200(US8987313, 30)
Affinity DataIC50: 170nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151186(US8987313, 8)
Affinity DataIC50: 170nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151192(US8987313, 29)
Affinity DataIC50: 190nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151190(US8987313, 21)
Affinity DataIC50: 190nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151198(US8987313, 49)
Affinity DataIC50: 190nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151188(US8987313, 16)
Affinity DataIC50: 200nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151185(US8987313, 5)
Affinity DataIC50: 230nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151186(US8987313, 8)
Affinity DataIC50: 240nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151197(US8987313, 42)
Affinity DataIC50: 250nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151189(US8987313, 18)
Affinity DataIC50: 260nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151196(US8987313, 39)
Affinity DataIC50: 260nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151187(US8987313, 11)
Affinity DataIC50: 300nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151188(US8987313, 16)
Affinity DataIC50: 300nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151191(US8987313, 25)
Affinity DataIC50: 300nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151192(US8987313, 29)
Affinity DataIC50: 310nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151201(US8987313, 31)
Affinity DataIC50: 330nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151190(US8987313, 21)
Affinity DataIC50: 340nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151199(US8987313, 24)
Affinity DataIC50: 340nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151193(US8987313, 32)
Affinity DataIC50: 350nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151200(US8987313, 30)
Affinity DataIC50: 360nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151195(US8987313, 36)
Affinity DataIC50: 370nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent

TargetCytochrome P450 3A4(Human)
Gilead Sciences

US Patent
LigandPNGBDBM151198(US8987313, 49)
Affinity DataIC50: 370nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/25/2015
Entry Details
Go to US Patent