Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 6636
LigandPNGBDBM142416(US8927738, 2-[2-(2-Furan-3-yl-1H-imidazol-4-yl)-et...)
Affinity DataIC50: 0.270nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142410(US8927738, 5,8-Dimethyl-2-[2-(2-thiophen-2-yl-1H-i...)
Affinity DataIC50: 0.340nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142414(US8927738, 5,8-Dimethyl-2-[2-(2-thiophen-2-yl-1H-i...)
Affinity DataIC50: 0.400nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142412(US8927738, 2-[2-(2-Furan-2-yl-1H-imidazol-4-yl)-et...)
Affinity DataIC50: 0.620nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142415(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-2-yl-1H-im...)
Affinity DataIC50: 0.630nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142413(US8927738, 2-[2-(2-Furan-3-yl-1H-imidazol-4-yl)-et...)
Affinity DataIC50: 0.650nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142409(US8927738, 2-[2-(2-Furan-2-yl-1-methyl-1H-imidazol...)
Affinity DataIC50: 0.75nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142417(US8927738, 2-[2-(2-Furan-2-yl-1H-imidazol-4-yl)-et...)
Affinity DataIC50: 0.970nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM50397979(US8927738, 5,8-Dimethyl-2-[2-(1-methyl-2-thiophen-...)
Affinity DataIC50: 1nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142406(US8927738, 2-[2-(2-Furan-2-yl-1-methyl-1H-imidazol...)
Affinity DataIC50: 1.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142411(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-2-yl-1H-im...)
Affinity DataIC50: 1.60nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142404(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-5-yl-1H-im...)
Affinity DataIC50: 3.10nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142407(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-4-yl-1H-im...)
Affinity DataIC50: 3.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142408(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-4-yl-1H-im...)
Affinity DataIC50: 3.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142418(US8927738, 5,8-Dimethyl-2-{2-[1-methyl-2-(5-methyl...)
Affinity DataIC50: 3.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142399(US8927738, 5,8-Dimethyl-2-[2-(2-phenyl-1H-imidazol...)
Affinity DataIC50: 4.20nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142396(US8927738, 8-Methoxy-5-methyl-2-[2-(2-phenyl-1H-im...)
Affinity DataIC50: 5.90nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142403(US8927738, 5,8-Dimethyl-2-[2-(2-thiazol-5-yl-1H-im...)
Affinity DataIC50: 6.5nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142402(US8927738, 5,8-Dimethyl-2-[2-(1-methyl-2-thiazol-2...)
Affinity DataIC50: 7.70nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142401(US8927738, 8-Methoxy-5-methyl-2-[2-(1-methyl-2-thi...)
Affinity DataIC50: 9nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142419(US8927738, 5,8-Dimethyl-2-[2-(1-methyl-2-thiazol-4...)
Affinity DataIC50: 11nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142420(US8927738, 2-{2-[2-(4-Fluoro-phenyl)-1H-imidazol-4...)
Affinity DataIC50: 12nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142405(US8927738, 5,8-Dimethyl-2-[2-(1-methyl-2-thiazol-5...)
Affinity DataIC50: 22nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142398(US8927738, 8-Ethyl-5-methyl-2-[2-(1-methyl-2-pheny...)
Affinity DataIC50: 23nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
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LigandPNGBDBM142400(US8927738, 5,8-Dimethyl-2-[2-(1-methyl-2-phenyl-1H...)
Affinity DataIC50: 45nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
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Date in BDB:
6/1/2015
Entry Details
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LigandPNGBDBM142397(US8927738, 8-Methoxy-5-methyl-2-[2-(1-methyl-2-phe...)
Affinity DataIC50: 79nMT: 2°CAssay Description:A PDE10A assay may for example, be performed as follows: The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2015
Entry Details
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