Report error Found 68 Enz. Inhib. hit(s) with all data for entry = 6587
Affinity DataIC50: 445nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 470nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 521nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 812nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 821nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 830nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.11E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.29E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.39E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.41E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.47E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.52E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.78E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.78E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.78E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.78E+3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.50E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.80E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+4nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 6nM ΔG°: -43.6kJ/mole IC50: 28nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 8nM ΔG°: -43.0kJ/mole IC50: 51.8nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 10nM ΔG°: -42.4kJ/mole IC50: 17.9nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 12nM ΔG°: -42.0kJ/mole IC50: 16.5nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 13nM ΔG°: -41.8kJ/mole IC50: 45.8nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 15nM ΔG°: -41.5kJ/mole IC50: 37nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 16nM ΔG°: -41.4kJ/mole IC50: 47.9nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 17nM ΔG°: -41.2kJ/mole IC50: 17.6nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 21nM ΔG°: -40.7kJ/mole IC50: 43.3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 28nM ΔG°: -40.1kJ/mole IC50: 32.8nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 29nM ΔG°: -40.0kJ/mole IC50: 34.7nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 30nM ΔG°: -39.9kJ/mole IC50: 65.7nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 31nM ΔG°: -39.8kJ/mole IC50: 43nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 32nM ΔG°: -39.8kJ/mole IC50: 19.8nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 32nM ΔG°: -39.8kJ/mole IC50: 46nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 32nM ΔG°: -39.8kJ/mole IC50: 54.9nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 38nM ΔG°: -39.4kJ/mole IC50: 41.5nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 49nM ΔG°: -38.8kJ/mole IC50: 83.9nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 60nM ΔG°: -38.3kJ/mole IC50: 76.7nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 66nM ΔG°: -38.1kJ/mole IC50: 55.3nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
Affinity DataKi: 69nM ΔG°: -38.0kJ/mole IC50: 100nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assays were performed in CHO cells expressing human CCR2B and Galpha ±16 coupling protein. All compounds were dissolved in DMSO a...More data for this Ligand-Target Pair
