Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 6585
TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140012(US8901310, Comparator B)
Affinity DataIC50: 0.350nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 0.526nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140015(US8901310, Comparator E)
Affinity DataIC50: 1.10nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140013(US8901310, Comparator C)
Affinity DataIC50: 1.10nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140015(US8901310, Comparator E)
Affinity DataIC50: 1.18nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140013(US8901310, Comparator C)
Affinity DataIC50: 1.22nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140014(US8901310, Comparator D)
Affinity DataIC50: 1.30nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140009(US8901310, Example 1 )
Affinity DataIC50: 1.31nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140016(US8901310, Comparator F)
Affinity DataIC50: 1.90nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140014(US8901310, Comparator D)
Affinity DataIC50: 2.06nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140017(US8901310, Comparator G)
Affinity DataIC50: 2.10nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140017(US8901310, Comparator G)
Affinity DataIC50: 2.13nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
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Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140019(US8901310, Comparator I)
Affinity DataIC50: 2.80nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140012(US8901310, Comparator B)
Affinity DataIC50: 4nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 4.20nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140018(US8901310, Comparator H)
Affinity DataIC50: 4.30nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140020(US8901310, Comparator J)
Affinity DataIC50: 4.58nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140016(US8901310, Comparator F)
Affinity DataIC50: 7nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140011(US8901310, Comparator A)
Affinity DataIC50: 7.10nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140018(US8901310, Comparator H)
Affinity DataIC50: 8.03nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140019(US8901310, Comparator I)
Affinity DataIC50: 9.12nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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LigandPNGBDBM19190((1S,2R,10S,11S,14R,15S,17S)-14,17-dihydroxy-14-(2-...)
Affinity DataIC50: 14.9nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140011(US8901310, Comparator A)
Affinity DataIC50: 36.4nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140010(US8901310, Example 2)
Affinity DataIC50: 42nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140010(US8901310, Example 2)
Affinity DataIC50: 60nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140010(US8901310, Example 2)
Affinity DataIC50: 79nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetInterleukin-6(Human)
Pfizer

US Patent
LigandPNGBDBM140020(US8901310, Comparator J)
Affinity DataIC50: 291nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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TargetGlucocorticoid receptor(Human)
Pfizer

US Patent
LigandPNGBDBM140021(US8901310, Comparator K)
Affinity DataIC50: 895nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
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LigandPNGBDBM140011(US8901310, Comparator A)
Affinity DataIC50: 1.00E+3nMAssay Description:The glucocorticoid receptor fluorescence polarization ligand binding (GRFP) assay is used to evaluate direct binding of testing compounds to full-len...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2015
Entry Details
Go to US Patent