Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with all data for entry = 6479
TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131030(US8835659, 11)
Affinity DataIC50: 1.84E+3nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
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TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM50336799(Suramin hexasodium | Germanin | suramin | 8,8'-[Ca...)
Affinity DataIC50: 2.62E+3nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent

TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131032(US8835659, 15)
Affinity DataIC50: 2.28E+4nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent

TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131031(US8835659, 13)
Affinity DataIC50: 3.67E+4nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent

TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131035(US8835659, 20)
Affinity DataIC50: 7.63E+4nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent

TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131034(US8835659, 19)
Affinity DataIC50: 1.92E+5nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent

TargetNAD-dependent protein deacetylase sirtuin-1(Human)
Ikerchem

US Patent
LigandPNGBDBM131033(US8835659, 16)
Affinity DataIC50: 2.74E+5nMpH: 8.0Assay Description:50 uM of substrate peptide (acetylated AMC-labeled peptide from p53 residues 379-382, RHKKAc, BioMol. Cat. #KI-177), 91 nM of human SIRT1 (full lengt...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/16/2015
Entry Details
Go to US Patent